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8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(furan-2-ylmethyl)-2-(4-methyl-1,4-diazepane-1-carbonyl)morpholine-4-carboxamide
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-oxobutane-1-sulfonamide
2-hydroxy-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(2-{4-[1-(propan-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-1-yl}ethyl)aniline
N-methyl-N-[2-(pyridin-2-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
3-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}phenol
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(diphenylmethyl)-N-[3-(methylsulfanyl)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
N-[(3R,4S)-4-cyclopropyl-1-[2-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
N-(2,3-dimethylpyridin-4-yl)-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
3-(2-chloro-5-methylphenyl)-1-ethyl-N,N-dimethyl-1H-1,2,4-triazol-5-amine
5-propyl-N-[3-(pyridin-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-4-methylphenol
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,4,4-trifluorobutanamide
3-{2-oxo-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-butyl-2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
1-(4-{4-methoxy-2-[4-(2-methoxyethyl)piperazine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
1-[3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperidine-4-carboxamide
N-cycloheptyl-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-[(4-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(3aR,6aS)-5-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
1-{5-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
N-{3-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(methyl)carbamoyl)amino]-4-methylphenyl}acetamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazine
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-{[5-(1-benzofuran-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
2,6-dimethyl-3-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
4-({[(4,6-dimethylpyridin-3-yl)methyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(3S,4R)-N,N-dimethyl-1-[4-(4-methylpiperazin-1-yl)benzoyl]-4-propylpyrrolidin-3-amine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3,4,7-trimethyl-1H-indole-2-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-methyl-2-{methyl[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]amino}acetamide
4-chloro-6-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
[1-(furan-3-ylmethyl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
3-(4-methyl-1,3-thiazol-5-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
1-(2H-1,3-benzodioxol-5-yl)-5-[2-(4-methylbenzenesulfonyl)ethyl]-1H-1,2,4-triazole
methyl 8-[(3,4-dimethylphenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-methyl-5-{[(3-methyl-5-propyl-1-benzofuran-2-yl)formamido]methyl}-1,2,4-oxadiazole-3-carboxamide