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2-methyl-4-(4-{[methyl(quinoxalin-2-ylmethyl)amino]methyl}phenyl)butan-2-ol
N-[(3R,4R)-3-hydroxy-1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-4-yl]pyrazine-2-carboxamide
3-[(2-fluoroethyl)sulfamoyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]benzamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[4-(furan-2-yl)pyrimidin-2-yl]-N,5-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
4-ethyl-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(2-methoxyethoxy)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
ethyl 1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H-imidazole-2-carboxylate
5,6-dimethyl-N4-[2-methyl-1-(pyridin-3-yl)propyl]pyrimidine-2,4-diamine
3-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
1-(3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-3-oxopropyl)azepan-2-one
methyl 3-benzamido-1-(oxolan-2-ylmethyl)-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
[(1-cyclopentylpiperidin-4-yl)methyl][(5-methylthiophen-2-yl)methyl](pyridin-3-ylmethyl)amine
6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(3-methoxyphenyl)-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(adamantan-1-yl)-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}acetamide
2-(3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carbonitrile
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
1-(furan-2-ylmethyl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]piperidine-4-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
1-(2-methoxyethyl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyrrolidine-3-carboxamide
3-{5-[1-(naphthalen-2-yloxy)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-[(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide
methyl 5-(2-aminopyridine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-(4-hydroxyphenyl)-N-[(3-methylpyridin-2-yl)methyl]benzamide
2-methyl-4-(2-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-tert-butyl-3-(oxan-4-yl)-1H-1,2,4-triazole
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
8-cyclopropanecarbonyl-2-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
2-(1H-1,3-benzodiazol-1-yl)-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]ethan-1-one
1-benzyl-4-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}piperazin-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
4-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
1-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)-4-(pyrrolidine-1-carbonyl)piperidine
N-[(3S,4R)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-(4-aminopyrimidin-2-yl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-hydroxy-2-(3-methylphenyl)-N-[3-(pyridin-4-yl)propyl]pyrimidine-5-carboxamide
(3aS,6aS)-2-[(2,5-dimethylthiophen-3-yl)sulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-[3-methyl-1-(naphthalen-1-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-ethyl-N-methyl-3-{[(5-methylpyrazin-2-yl)methyl]sulfamoyl}benzamide
6-cyclopropyl-N-[1-(3,4,5-trimethoxyphenyl)ethyl]pyrimidin-4-amine
4-(2-methyl-1H-imidazol-1-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}butan-1-one
4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(2-phenylethyl)piperidine-1-carboxamide
4-(5-tert-butyl-1H-pyrazol-3-yl)-1-[(2-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one