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1-[7-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4-methylphenyl)propan-1-one
9-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(3-fluorophenyl)-1-methyl-3-{2-[3-(3-methylbutanoyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-[({5-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
4-methyl-3-oxo-N-[3-(phenylsulfanyl)propyl]-3,4-dihydroquinoxaline-2-carboxamide
3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(4-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
1-(2-methoxyethyl)-3-(3-methoxyphenyl)-3-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
1-cyclopropanecarbonyl-N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
1-(4-{4-azaspiro[2.5]octan-4-ylmethyl}-2-methoxyphenoxy)-3-(azepan-1-yl)propan-2-ol
1-(cyclohexylmethyl)-5-[(3-hydroxy-2,2-dimethylpropyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
5-butyl-6-methyl-N4-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidine-2,4-diamine
4-{[(2,3-dihydro-1H-inden-2-yl)(methyl)amino]methyl}-1H-pyrazole-3-carboxylic acid
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-N-(pyridin-3-ylmethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[6-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]piperidine-4-carbonitrile
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-8-methylimidazo[1,2-a]pyridine-2-carboxamide
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
methyl 4-{[7-(2-hydroxy-1-phenoxypropan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
N-[(3R,4R)-3-hydroxy-1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl]pyridine-3-carboxamide
3-(azepane-1-carbonyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-chloro-2-[1-(1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
1-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
3-({[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
6-(pyrrolidin-1-ylmethyl)-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1,4-oxazepan-6-ol
(3R,4R)-1-[(2,3-difluoro-4-methylphenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
9-[2-(dimethylamino)propanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(cyclohexylsulfanyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 4-(2-{[cyclohexyl(prop-2-yn-1-yl)amino]methyl}-8-methylquinazolin-4-yl)piperazine-1-carboxylate
7-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-2-oxa-7-azaspiro[4.5]decane
2-(3-{[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenoxy)ethan-1-ol
3-cyclopentyl-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
6-(benzyloxy)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(oxan-4-ylmethyl)-1,4-diazepan-2-one
1-(1H-indazol-4-yl)-3-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]urea
3-[3-(azepane-1-carbonyl)phenyl]-1-(2-phenoxyethyl)urea
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(3-methylpyridin-4-yl)methyl]propanamide
6-fluoro-2-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}quinolin-4-ol
N-[(8-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]benzamide
N-(2-methoxyethyl)-1-[1-(4-methylpent-3-en-1-yl)piperidin-4-yl]piperidine-3-carboxamide
3-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-3-(3-fluorophenyl)-1-methylpyrrolidine-2,5-dione
9-[(2E)-3-phenylprop-2-en-1-yl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
N-[2-(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxolane-2-carboxamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(5-methylhex-5-en-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one