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2-ethyl-4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
5-{[2-(2-chlorophenyl)ethyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}thiomorpholine
1-(4-chlorophenyl)-N-{[1-(3-methylfuran-2-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
S-[2-(ethanesulfonyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]-3-hydroxybutane-1-sulfonamido
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-(1,3-thiazol-2-ylmethyl)piperidin-3-ol
N-[3-(oxolan-3-yl)propyl]-2-(4-propanoylphenoxy)acetamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazine
1-cyclohexyl-4-(1H-pyrazol-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
methyl (2S,4S)-4-(2-ethoxypyridine-3-amido)-1-methylpyrrolidine-2-carboxylate
N-({1-[(3-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)piperidine-4-carboxamide
2-methyl-4-{4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]phenyl}butan-2-ol
1-(2-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
1-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}-1,3-diazinane-2,4-dione
3-phenyl-1-[4-(quinolin-6-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-1-ol
2-[4-(1-methyl-1H-pyrrole-2-carbonyl)morpholin-3-yl]-1-(thiomorpholin-4-yl)ethan-1-one
(2R,6R)-4-(pent-2-yn-1-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-(2-fluorophenyl)-N-methyl-N-[2-(piperidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
{[4-(5-chloro-3-methyl-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
4-(4-methyl-1H-pyrazol-1-yl)-1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidine-4-carboxylic acid
1,3-dimethyl 5-{[2-(2-hydroxyethyl)piperidine-1-carbonyl]amino}benzene-1,3-dicarboxylate
N-[3-(methylsulfanyl)propyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(4-methylphenyl)ethyl]benzamide
N-(1H-indol-6-ylmethyl)-2,5,6-trimethylpyrimidin-4-amine
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
10-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-ethoxypropanamide
3-(4-chlorophenyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(2-methyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
2-methyl-7-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
3-[4-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]piperidine-1-carboxamide
5-(2-butoxy-5-methylphenyl)pyridin-3-amine
(1R,7S)-3-cycloheptyl-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-ethyl-N-[(1R,2R)-2-hydroxycyclohexyl]-4-methyl-N-propyl-1H-pyrazole-5-carboxamide
(3S)-4-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1-ethyl-3-methylpiperazin-2-one
(2S,4S)-4-amino-1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}piperidin-4-amine
1-[(3-fluorophenyl)methyl]-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
N-(dicyclopropylmethyl)-6-(3-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methoxy-3-(morpholin-4-yl)benzamide
N-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-(morpholin-4-yl)-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
2-cyclopropyl-5-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]pyrimidin-4-ol
N-cyclohexyl-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one