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(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-amine
2,3-dimethyl-6-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-(2-hydroxyethyl)piperidine-4-carboxamide
2-(4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}morpholin-2-yl)ethan-1-amine
N-[1-(6-methylpyridin-2-yl)propan-2-yl]-5-propyl-1,3,4-oxadiazol-2-amine
1-(4-ethylpiperazin-1-yl)-3-[3-(pyrrolidin-1-ylmethyl)phenoxy]propan-2-ol
6-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-benzothiazole
N-[2-(4-phenylpyrimidin-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-methoxy-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(pyridin-4-yl)propan-1-one
5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazole
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(3-methoxyphenyl)ethyl]propanamide
7-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(4-{[2-(4-fluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-phenoxypropanamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-propylpiperidine
(3aR,7aS)-5-methyl-2-[2-(morpholin-4-yl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
N-[4-(6-hydroxy-1,4-oxazepane-4-carbonyl)phenyl]ethane-1-sulfonamide
1-[(4-methoxyphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
ethyl 4-[(4-methoxyphenyl)methyl]-1-(pyridine-3-carbonyl)piperidine-4-carboxylate
4-({1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)benzoic acid
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(3,3,5,5-tetramethylcyclohexyl)propanamide
4-(azepane-1-carbonyl)-2-(2-cyclopropylpyrimidin-5-yl)-6-methylquinoline
3-(4-chlorobenzoyl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyridin-4-yl)ethan-1-one
1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N-(2-hydroxyethyl)piperidine-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-3-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperazin-2-one
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
ethyl 1-({2-[butyl(methyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)piperidine-4-carboxylate
(3S,4R)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-fluoro-2-methoxy-N-[1-(2-methoxyphenyl)ethyl]-N-methylbenzamide
1-methyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]pyrrolidine-3-carboxamide
1-{2-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}azepan-2-one
N-methyl-N-(3-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-3-oxopropyl)methanesulfonamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
4-[(2,2-difluoroethyl)sulfamoyl]-N-(furan-3-ylmethyl)benzamide
1-(1-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
5-[(2,5-dimethoxyphenyl)methyl]-4-(5-methylfuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-(4-chlorophenoxy)-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-4-carboxamide
2-[(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)methyl]benzonitrile
5-(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
7-fluoro-N-(1-methylpiperidin-4-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
(2R,3R)-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol