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N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethylthiophene-3-carboxamide
2-{1-cyclohexyl-4-[(2,4-dimethoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethylpyrimidine-5-carboxamide
N-{3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-2-fluorobenzamide
N3-(butan-2-yl)-1-cyclopentyl-N5-(cyclopropylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-benzyl-1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
1-(4-{[(1H-indol-4-ylmethyl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
1-[(1-benzyl-1H-imidazol-5-yl)methyl]azepan-2-one
5-{1-[2-(2,6-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
2-(2-hydroxypropyl)-9-(2-hydroxypyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(4-chlorophenyl)acetyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
(3R,4S)-4-cyclopropyl-1-(6-cyclopropylpyrimidin-4-yl)pyrrolidin-3-amine
3-{imidazo[1,2-a]pyridin-2-yl}-N-[(1-methanesulfonylpiperidin-3-yl)methyl]propanamide
(1R,5S)-6-methyl-3-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-phenyl-1,3-thiazol-4-yl)-1-[4-(3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethan-1-one
5-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
N,3,5,7-tetramethyl-N-(oxan-2-ylmethyl)-1H-indole-2-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(3-phenoxypropyl)acetamide
2-[(1-{1-[(5-methyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]-2-azaspiro[4.4]nonane
1-(diethylamino)-3-[2-methoxy-4-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N4-[(1-ethyl-1H-imidazol-2-yl)methyl]-N2,N2,N4,5,6-pentamethylpyrimidine-2,4-diamine
1-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
N-(1-carbamoylcyclopentyl)-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
methyl 3-{6-[(3-methoxyphenyl)methoxy]-2-oxo-4-(4-oxo-4-phenylbutanoyl)-1,4-diazepan-1-yl}propanoate
(2S,4S)-N-ethyl-1-methyl-4-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanamido}pyrrolidine-2-carboxamide
1-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-3-methylpiperidine-3-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
7-(3-methoxypropanamido)-1-methyl-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
methyl 3-(2-chlorobenzenesulfonamido)-5-{[2-(thiophen-3-yl)acetamido]methyl}benzoate
1-[2-oxo-2-(4-phenyl-1,4-diazepan-1-yl)ethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-(4-chloro-3-methoxyphenyl)-2-{[(2,5-difluorophenyl)methyl]amino}acetamide
2-[6-(2-methoxyphenyl)pyridazin-3-yl]-N,N-dimethylaniline
(4aR,8aR)-2-methanesulfonyl-7-{[2-(propylamino)pyrimidin-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidin-2-yl]pyridine
3-(methoxymethyl)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2-oxopropanamide
5-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}pyridin-2-amine
(3S,5R,9R)-11-[(4-chlorophenyl)methyl]-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-[1-(3-cyano-4,6-dimethylpyridin-2-yl)piperidin-3-yl]-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
2-{4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}ethan-1-ol
N-[(2-methylphenyl)(pyridin-4-yl)methyl]-1-propylpiperidin-4-amine
2-methoxy-4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
N-methyl-5-{[methyl(propan-2-yl)amino]methyl}-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(oxan-4-yl)piperazine
(4aS,8aR)-6-[(4,5-dimethylfuran-2-yl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
ethyl[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](oxan-4-ylmethyl)amine
3-methoxy-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-N-methyl-7-oxo-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(2-methylfuran-3-carbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid