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1-{3-oxo-3-[3-(2-phenylacetyl)piperidin-1-yl]propyl}-1,2-dihydropyridin-2-one
4-fluoro-N-(2-{[3-(trifluoromethyl)-1H-pyrazol-5-yl]formamido}ethyl)benzamide
3-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[2-(pyridin-2-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
(2S,4S)-4-amino-N,N-diethyl-1-(9H-purin-6-yl)pyrrolidine-2-carboxamide
1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-4-(pyridin-3-yl)piperazine
N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
diethyl({[3-(1,2,3,6-tetrahydropyridine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
8-fluoro-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]quinoline-2-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
(2S,4S)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N,1-bis[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-(2-methoxyethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
5-(azocane-1-carbonyl)-1-[(3-methoxyphenyl)methyl]piperidin-2-one
3-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
7-[(4-fluorophenyl)methyl]-2-{[5-(hydroxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-(4-{[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}phenyl)ethan-1-one
N-(4-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}phenyl)acetamide
5-[4-(aminomethyl)piperidin-1-yl]-2-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,3-dihydropyridazin-3-one
1-[2-(isoquinolin-5-yl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
5-chloro-N-[(1-propyl-1H-pyrazol-4-yl)methyl]pyridine-2-carboxamide
4-{2-methyl-1H-imidazo[4,5-b]pyridin-6-yl}-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-methoxy-1,2-dimethyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1H-indole-3-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-(1H-pyrrole-2-carbonyl)piperidin-3-ol
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2-methylphenol
2-(3-methoxypropyl)-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[(4-phenoxyphenyl)methyl]propanamide
1-[1-(azepane-1-sulfonyl)piperidin-3-yl]-2-phenylethan-1-one
2-ethyl-8-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
8-cyclopentyl-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
N-cyclohexyl-2-{6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-oxoacetamide
1-{3-[({imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
N-cyclopropyl-1-[1-(4-methylpyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
4-{furo[3,2-c]pyridin-4-yl}benzamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-1-yl]acetamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[(3,5-dimethoxyphenyl)methyl]acetamide
3-(3-fluorophenyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-(diethylamino)-3-(2-methoxy-4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenoxy)propan-2-ol
5-chloro-2-(3-ethylmorpholine-4-carbonyl)-3-phenyl-1H-indole
N-methyl-N-{2-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N-(2-methylpropyl)-2-oxoacetamide
N-(5-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}pyrimidin-2-yl)benzenesulfonamide
N-({7-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
2-methoxy-6-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-(oxan-3-yl)urea
6-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]pyrazine-2-carboxamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(thiophen-3-yl)-1H-pyrazol-1-yl]acetamide