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5-[(4-hydroxypiperidin-1-yl)methyl]-N,N-dipropyl-1,2-oxazole-3-carboxamide
2-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}-4-methoxyphenol
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[1-(hydroxymethyl)cyclopropyl]acetamide
2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]acetamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
4-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)thiomorpholine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-pyrazole-4-carboxamide
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
1-(1-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
2-(ethoxymethyl)-N-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[3-(4-hydroxypiperidin-1-yl)propyl]-5-methyl-5-phenylpiperidin-2-one
1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidine-1-sulfonyl)piperazine
(3S)-1-[6-ethyl-2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
(3S,9aR)-8-(4-chlorobenzenesulfonyl)-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-fluorophenyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidine
1-(4-benzylpiperazin-1-yl)-3-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propan-1-one
2-[(1S,5R)-6-(5-acetylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-(1-ethylpiperidin-4-yl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]acetamide
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(methylsulfanyl)phenyl]urea
N-[(5-chlorothiophen-2-yl)methyl]-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
2-{[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-4-oxo-1,4-dihydroquinoline-6-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
2-[benzyl({4-[(thiophen-2-ylmethyl)amino]quinazolin-2-yl}methyl)amino]ethan-1-ol
N-{[(3S,4S)-3-hydroxy-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]methyl}-2-methoxybenzamide
N-(2,6-dimethylphenyl)-2-[2-(2-methyl-1H-imidazol-1-yl)propanamido]benzamide
2-(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-4-methyl-1H-1,3-benzodiazole
5-methoxy-3-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)-1H-indazole
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxylic acid
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]acetamide
6-(4-cyclopentylpiperazin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
6-methoxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,3-dimethyl-1-benzofuran-2-carboxamide
2-{[7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-5-methoxyphenol
4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine-1-sulfonamide
1-{1-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
butyl (4aS,7aR)-6,6-dioxo-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-cyclohexylurea
4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-[3-(methylsulfanyl)propyl]benzamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-[ethyl(methyl)amino]propan-1-one
(4aR,8aS)-6-{[3-(benzyloxy)phenyl]methyl}-1-(2-methoxyethyl)-decahydro-1,6-naphthyridin-2-one
4-fluoro-N-(2-{[2-(methylamino)pyrimidin-5-yl]formamido}ethyl)benzamide
(1R,2S)-1-[(4-cyclopentylpyrimidin-2-yl)amino]-2,3-dihydro-1H-inden-2-ol
3-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}pyrazine-2-carbonitrile
1-{2-methyl-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]phenyl}imidazolidin-2-one
1-(9H-purin-6-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
dimethyl[2-(2-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}phenoxy)ethyl]amine
4,6-dimethyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-2-amine
4-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1,2-dihydroquinolin-2-one
1-[2-(dimethylamino)-4-{[(5-methylfuran-2-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one