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N-(1-hydroxy-2-methylpropan-2-yl)-5-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-[1-(1H-indole-5-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(2R,3R,6R)-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl})(propan-2-yl)amine
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]oxane-4-carboxamide
propyl 4-(2-ethoxy-2-oxoethyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
2-[4-(cyclohexylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2,6-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-hydroxypropyl)piperidine-4-carboxamide
(3S)-3-ethyl-N-(2-phenylphenyl)morpholine-4-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxylate
1-[(diethylcarbamoyl)methyl]-N-[2-(furan-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-4-yl}thiomorpholine
2-(4,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
2-methyl-6-[2-(3-phenylpropyl)morpholine-4-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-(pyridin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
2-(1H-pyrrol-1-yl)-5-(2,3,4-trimethoxyphenyl)pyridine
methyl[(2-methyl-1,3-oxazol-4-yl)methyl][(4-phenoxyphenyl)methyl]amine
(3R,4S)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(3-methoxyphenyl)pyrrolidin-3-amine
N-[(4-phenylphenyl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
2-{[(4-fluorophenyl)methyl][3-(methylsulfanyl)propyl]amino}butan-1-ol
6-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
7-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-(2,5-dimethyl-3-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}-1H-pyrrol-1-yl)acetamide
N-(1-benzylpiperidin-4-yl)-2-ethyl-6-methyl-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-[4-(benzyloxy)piperidine-1-carbonyl]-2-(methylsulfanyl)pyridine
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]methylamine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,3-dihydro-1H-indene-1-carboxamide
2-(cyclopropylmethyl)-N-(3-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
7-(3-chlorophenyl)-4-(piperidine-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-cyclopropyl-5-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-methyl-6-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-{4-chloro-3-[2-(cyclohex-3-en-1-yl)-1H-imidazol-1-yl]phenyl}-2-methoxyacetamide
1-(2-amino-4-methylpyrimidine-5-carbonyl)-4-methylpiperidine-4-carbonitrile
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]benzamide
3-methoxy-N-(1-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
N-[1-(3-chlorophenyl)cyclopropyl]-2-(propan-2-yloxy)propanamide
[(2,3-dichlorophenyl)methyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-2-oxo-1-phenylpyrrolidine-3-carboxamide
(4aS,7aR)-1-[(2-chlorophenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(cyclopropylmethyl)-5-(3-methylthiophen-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[4-(3-cyanophenyl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]-2-methoxyacetamide
1-cyclopentyl-4-{[methyl({5-methylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}pyrrolidin-2-one
2-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}pyridine-4-carbonitrile
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
(3aR,6aR)-2-cyclopropanecarbonyl-N-(3-phenylpropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(5-acetylthiophen-3-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
1-(furan-3-carbonyl)-3-[2-(methylsulfanyl)benzoyl]piperidine