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1-cyclohexanecarbonyl-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
3-(5-methylfuran-2-yl)-1-[(4-methylphenyl)methyl]-5-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-1,2,4-triazole
2-(2-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}phenoxy)ethan-1-ol
3-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}quinoline
1-ethyl-3-(2-methyl-1,3-benzothiazol-6-yl)-1-[2-(1H-pyrazol-1-yl)ethyl]urea
N,N-dimethyl-3-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}piperidine-1-carboxamide
N-{2-[1-(2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperidin-4-yl]ethyl}acetamide
9-[(3-chloro-4-fluorophenyl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)urea
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-[(2R,3R)-1'-[(4-hydroxy-3,5-dimethylphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
5-{[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-thiadiazol-2-amine
4-methyl-7-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-2H-chromen-2-one
2-(3-methoxy-4-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(2-methoxyethyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
2-acetyl-8-(2-cyanobenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(1S,3R)-3-amino-N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}cyclopentane-1-carboxamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3R,4S)-4-cyclopropyl-1-[(2,5-dimethylthiophen-3-yl)sulfonyl]pyrrolidin-3-amine
1-{5-[(dimethylamino)methyl]-1,3,4-oxadiazole-2-carbonyl}-N,N-dimethylpyrrolidin-3-amine
N-[2-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)ethyl]acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,3-thiazole-4-carbonyl)pyrrolidine-3-carboxylic acid
3-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(dimethylamino)methyl]-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]azepan-4-ol
N4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-6-(morpholin-4-yl)pyrimidine-2,4-diamine
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-amine
(3R,4R)-1-(6,8-difluoro-2-methylquinolin-4-yl)-4-ethylpiperidine-3,4-diol
1-(2-methoxy-2-methylpropyl)-2-(2-methylphenyl)-1H-imidazole
2-[3-(5-chlorothiophen-2-yl)-1H-pyrazol-1-yl]-N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
5-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
[3-(2-ethyl-1H-imidazol-1-yl)propyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
6-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-benzothiazole
ethyl 2-{[5-(2,5-dihydro-1H-pyrrol-1-ylmethyl)pyrimidin-2-yl](methyl)amino}acetate
1-(2-phenoxyethyl)-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
1-(1-cyclopentylpiperidine-3-carbonyl)-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
N-(5-phenyl-1,3,4-thiadiazol-2-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
2-(2,3-difluorophenoxymethyl)-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-1,3-oxazole-4-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopentanecarboxamide
[(1-cyclopentylpiperidin-3-yl)methyl][(4-methyl-1H-imidazol-2-yl)methyl][2-(piperidin-1-yl)ethyl]amine
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-[(2-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropan-1-amine
1-(3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}piperidin-1-yl)ethan-1-one
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidin-2-amine
1-(cyclopropylmethyl)-5-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[5-(4-chlorophenyl)-1,2-oxazol-3-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
(3R,4R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-3,4-dimethylpyrrolidin-3-ol