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1-[2-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
{4-[(1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl)methyl]phenyl}methanol
1-[(2,3-dichlorophenyl)methyl]-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3S,5S)-5-(diethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
(2-{2-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-[(dimethylamino)methyl]-1,3-thiazole-4-carboxamide
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
8-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(5-methyl-4-{[(4-methyl-1,3-oxazol-5-yl)formamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-ethoxy-4-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
(3S)-1-benzyl-N-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-amine
3-(oxolan-3-yl)-5-[2-(1H-1,2,4-triazol-1-yl)phenyl]-1,2,4-oxadiazole
2-cyclopropyl-8-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
propyl 2-[(3-cyanophenyl)methyl]-2,7-diazaspiro[4.5]decane-7-carboxylate
4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)-N-(1H-indazol-5-yl)piperazine-1-carboxamide
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-(1H-imidazol-2-ylmethyl)urea
4-{3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanoyl}-1-phenylpiperazin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-ol
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-3-ol
4-(4-methylpiperazin-1-yl)-6-(1H-pyrazol-3-yl)pyrimidin-2-amine
N-methyl-4-oxo-4-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]butanamide
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]urea
3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
7-[(5-methylpyrazin-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-(phenylsulfanyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-(dimethyl-1,2-oxazol-4-yl)-5-[1-(furan-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyridine-3-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1-ethylpiperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-5-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-imidazole
5-(3,4-dimethylphenoxymethyl)-N-[2-(4-methylpiperazin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
(3S)-3-amino-3-{[(3-chlorophenyl)methyl](propyl)carbamoyl}propanoic acid
[1-(1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
N-[2-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclobutanecarboxamide
2-methoxy-5-(2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)phenol
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
N-[(2-{4-[3-(4-methoxyphenyl)propanamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]furan-3-carboxamide
1-(3,4-difluorophenyl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
2-chloro-4-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}phenol
2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-N-methylpyridine-4-carboxamide
2-amino-N-methyl-6-(propan-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-4-carboxamide
1-{[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]methyl}pyrrolidin-2-one
(2S,3R)-3-hydroxy-2-[4-phenyl-5-(5-propylfuran-2-yl)-1H-imidazol-1-yl]butanamide
8-[4-(3-fluorophenyl)benzoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-(2-methylprop-2-en-1-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
1-{2-[3-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
7-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-benzofuran-2-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(4-methoxyphenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-[2-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
5-(2,6-dichlorophenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole