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2-phenyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
N-benzyl-N-(cyclobutylmethyl)-4-propylpyrimidine-5-carboxamide
N-(1-carbamoylcycloheptyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
1-[(4-chlorophenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)piperidine-3-carboxamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-1H-pyrrole-2-carboxamide
N-[1-(4-methanesulfonylphenyl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-({1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-[5-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)-1H-pyrazol-3-yl]ethan-1-one
6-[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)amino]-N-ethylpyridine-3-carboxamide
5-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
3-chloro-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
N-[(3R,4S)-1-(cyclobutylmethyl)-4-cyclopropylpyrrolidin-3-yl]-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(3S,4R)-N,N-dimethyl-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
4-[(2-fluoro-4-methoxyphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
1-[3-({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
(2S)-2-[(1-cyclopentylpiperidin-4-yl)formamido]-3-(4-hydroxyphenyl)propanamide
5-(2-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-methyl-1-{3-oxo-3-[4-(pyridin-4-yl)piperidin-1-yl]propyl}-1,2-dihydropyridin-2-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
5-[1-(2,3-dimethoxybenzoyl)piperidin-4-yl]-3-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione
8-fluoro-3-[1-(pyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
N-[(2-methoxyphenyl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
N-(2-methanesulfonylethyl)-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
4-[3-(2-ethyl-3-oxopiperazine-1-carbonyl)phenoxy]-N,N-dimethylpiperidine-1-sulfonamide
N-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-4-yl}methanesulfonamide
3-methoxy-2-{[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
2-(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methyl-1,2-oxazole-5-carboxamide
N-(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
7-(3-chlorophenyl)-4-(1-ethyl-1H-pyrazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(3-hydroxyphenyl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
(2S,4S)-4-[(1-ethylpiperidin-4-yl)amino]-1-(naphthalen-2-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(2-{4-[2-(phenylsulfanyl)acetamido]-1H-pyrazol-1-yl}acetyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
1-methyl-3-(4-phenylbenzoyl)piperidine
1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
5-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
methyl (2S)-3-(1H-imidazol-4-yl)-2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propanoate
N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
1-({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)-4-methylpiperidine-4-carbonitrile
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}oxolane-3-carboxamide
3-(2-ethylbutyl)-8-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}pyrimidine
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)cyclopentanecarboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(2-methoxyphenyl)ethan-1-one
N-methyl-2-(thiophen-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[4-(3,3-diphenylpiperidin-1-yl)-4-oxobutan-2-yl]acetamide
2-[1-(propan-2-yl)-4-(pyridin-4-ylmethyl)piperazin-2-yl]ethan-1-ol