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2-ethoxy-3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}pyridine
N-({4-[benzyl(ethyl)amino]quinazolin-2-yl}methyl)cyclohex-3-ene-1-carboxamide
4-({2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}sulfonyl)morpholine
{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
2-(1-propylpiperidin-4-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
(4aR,8aR)-2-methanesulfonyl-7-(1,3-thiazol-4-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
4-methoxy-6-[4-(2-propoxyethyl)piperazin-1-yl]pyrimidine
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,5-thiadiazole-3-carboxamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
N-(2,3-dihydro-1-benzofuran-3-yl)-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
(4aS,7aR)-1-[3-(1H-indol-3-yl)propanoyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(3-hydroxy-4-methoxyphenyl)methyl]-6-methyl-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
3-chloro-4-{[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
1-(3-methylpyridin-2-yl)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(2-phenylethyl)piperidine-3-carboxamide
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]pyridine-2-carbonitrile
4-{3-[2-(3-methoxyphenyl)-1H-imidazol-1-yl]propoxy}-1-methylpiperidine
2-amino-4-(2-phenylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(6-fluoropyridin-3-yl)urea
4-chloro-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
4-{1-cyclohexyl-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}butanoic acid
N-[2-(diethylamino)ethyl]-2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-ethylacetamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(4-methylpiperazine-1-carbonyl)pyrazine
4-methyl-6-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-2-amine
3-{1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]piperidin-3-yl}propan-1-ol
N-(oxolan-2-ylmethyl)-N-propyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
N-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1-azabicyclo[2.2.2]octan-3-amine
N-methyl-N-(quinolin-5-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-(6-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-2-yl)ethan-1-ol
[(3R,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(morpholine-4-carbonyl)piperidin-3-yl]methanol
2-oxo-N-(2-phenylethyl)-6-(propan-2-yl)-N-propyl-1,2-dihydropyridine-3-carboxamide
dimethyl(3-{2-[1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
2-(pent-4-enoyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
methyl 3-acetamido-1-methyl-5-{[(3-methylphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-2-azaspiro[4.4]nonan-3-one
2-methyl-5-({4-phenyl-5-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1,3,4-oxadiazole
3-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)propanamide
N-(1-{7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
1-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]azepane
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-hydroxy-3-(3-methoxyphenoxy)propyl]urea
3-{1-[(2-chlorophenyl)methyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-4-methoxyphenol
N-methyl-2-(2-oxopiperidin-1-yl)-N-[(4-phenoxyphenyl)methyl]acetamide
1-[4-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)thiophen-2-yl]ethan-1-one
5-{2-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-oxoethyl}pyrrolidin-2-one
(2-oxo-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)urea
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-[3-(propan-2-yloxy)propyl]acetamide