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3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyridazine
2-(3-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
(3R,4S)-1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-4-cyclopropylpyrrolidin-3-amine
1-(3-phenylpropyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,4-diazepane
(3R,4S)-1-(2-fluoro-5-methylbenzenesulfonyl)-4-propylpyrrolidin-3-amine
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-5-methoxyphenol
(2-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)dimethylamine
8-(cyclohex-3-en-1-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3S,5S)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-3-methyl-1H-pyrazole-5-carboxamide
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
3-[(4-fluorophenyl)formamido]-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]propanamide
2,3-dimethyl-6-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
4-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-3-yl]-5-phenyl-2-(pyridin-4-yl)pyrimidine
4,6-dimethyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(5-methyl-4-{[2-(pyridin-2-ylsulfanyl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]cyclobutanecarboxamide
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
2-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
N-{[2-chloro-5-(trifluoromethyl)phenyl]methyl}-4-methylpiperidine-4-carboxamide
2-chloro-4-({[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]ethan-1-one
dimethyl({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}sulfamoyl)amine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]propanamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[2-(propan-2-yloxy)ethyl]pyridin-2-amine
(4aS,7aR)-1-[(2,4-difluorophenyl)methyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
N-[(4-phenyloxan-4-yl)methyl]-6-(thiophene-3-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
8-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-ethyl-N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[furan-2-yl(phenyl)methyl]-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-benzyl-2-(2,5-dioxoimidazolidin-1-yl)-N-[(1R,2R)-2-hydroxycyclohexyl]acetamide
3-({2-[1-(oxane-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-[2-(4-fluorophenyl)morpholine-4-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
1-cyclohexyl-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-[(thiophen-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[1-(1-aminocyclobutanecarbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-pentanamidobenzamide
2-{3-[(3,4-dimethoxyphenyl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}ethan-1-ol
5-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-2-methyl-1H-1,3-benzodiazole
N-ethyl-N-(2-methoxyethyl)-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
4-{1-[(1-hydroxycyclohexyl)methyl]-1H-imidazol-2-yl}benzoic acid
4-[4-(3-methylthiophene-2-carbonyl)piperazin-1-yl]quinazoline
1-(2-phenylethyl)-8-[(2E)-3-phenylprop-2-en-1-yl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-9-(5-propyl-1,3,4-oxadiazol-2-yl)-3,9-diazaspiro[5.6]dodecane
4-methyl-1-(naphthalene-1-carbonyl)-1,4-diazepan-5-one
2-{[(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
N-{1-[4-(6-methyl-9H-purin-9-yl)phenyl]ethyl}acetamide
1-methyl-N-[3-(morpholin-4-yl)propyl]-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide