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(2R,3R,6R)-3-(3,5-difluorophenyl)-5-propyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(methylsulfamoyl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
4-(4-ethoxy-3-methylphenyl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]butanamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-N-cyclopentyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
3-(1,2-oxazolidin-2-yl)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
3-fluoro-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzene-1-sulfonamide
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-cyclopentyl-4-[4-(morpholine-4-carbonyl)pyridin-2-yl]-1,4-diazepane
5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
[(1-ethyl-1H-pyrazol-4-yl)methyl]({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(1,2-oxazol-5-ylmethyl)acetamide
3-(5-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-1-(pyrrolidin-1-yl)propan-1-one
1-(propan-2-yl)-2-({3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-imidazole
(1S,5R)-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-chlorothiophen-2-yl)-4-methoxypyrimidine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(3-methoxyphenoxy)ethyl]-N-methylbenzamide
(3S,4S)-1-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
[(4-ethoxyphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-{[(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
4-{3-[4-(4-chlorophenyl)-4-hydroxypiperidine-1-carbonyl]piperidin-1-yl}-2-(2,2-dimethyloxan-4-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
N-[3-(2-methoxyethoxy)phenyl]-3-(pyrimidin-4-yl)piperidine-1-carboxamide
methyl 4-[({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)carbamoyl]butanoate
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-hydroxy-4-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
3-cyclopentyl-N-[2-(1-methylpiperidin-3-yl)ethyl]propanamide
(4aS,8aR)-6-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-[(5-fluoro-1H-indol-2-yl)methyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
3-{1-[5-(methoxymethyl)furan-2-carbonyl]azetidin-3-yl}pyridine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(5-methylthiophen-2-yl)methyl]benzamide
2-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
1-{4-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
N-cyclopropyl-1-methanesulfonyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
2-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1,3-benzoxazole
ethyl 1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine-3-carboxylate
1-[5-({[5-(hydroxymethyl)furan-2-yl]methyl}amino)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl]piperidin-4-ol
3-methyl-1-{1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}butan-1-ol
1-methyl-3-(3-{4-[(1,3-thiazol-2-ylmethyl)amino]piperidin-1-yl}phenyl)imidazolidin-2-one
N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-2-(pyrrolidin-3-yl)benzamide
N-[2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-1-phenylcyclopropane-1-carboxamide
2-butyl-5-(1,2-oxazolidine-2-carbonyl)-1,3-benzoxazole
2-methoxy-6-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
8-(2-methoxy-4-methylbenzenesulfonyl)-2-methyl-2,8-diazaspiro[4.5]decane
N-[(1-benzylpyrrolidin-3-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)-N-methylacetamide
2,4,7-trimethyl-3-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
1-methyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-methyl-6-(pyrrolidine-1-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetamide
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine