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2-amino-6-(4-hydroxyphenyl)-4-(1H-indol-3-yl)pyridine-3-carbonitrile
1-(1'-{[6-(dimethylamino)pyridin-3-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
2-[3-(1-butyl-1H-1,2,4-triazol-5-yl)propyl]-5-(4-fluorophenyl)-2H-1,2,3,4-tetrazole
2-methyl-6-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-[(1S,2R)-2-[(1-acetylpiperidin-4-yl)amino]cyclobutyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
N-(furan-3-ylmethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}-4-(2,5-dimethoxyphenyl)phenol
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(5-methylpyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{4-[(benzylsulfamoyl)amino]phenyl}pyridine-3-carboxamide
3-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]-4-(pyridin-2-ylmethyl)piperazin-2-one
7-fluoro-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-2-methylquinoline-4-carboxamide
N-[(2-fluorophenyl)methyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
4-({5-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(1-methylpiperidin-4-yl)piperazine
2-(2-aminoethyl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}quinazolin-4-amine
4-hydroxy-N-[2-(1H-imidazol-4-yl)ethyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N,N-dimethylacetamide
5-methyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
(3aS,6aR)-5-(3-chloropyridin-2-yl)-3-cyclopentyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(4-tert-butylphenyl)-5-methylpyrimidin-4-amine
(1S,5R)-6-(dimethyl-1,3-oxazole-5-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(3,4-dimethylphenyl)-1-(furan-3-carbonyl)piperidin-3-amine
3-[({1-[(3,4-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(pyridine-4-carbonyl)piperidin-3-yl]piperazine
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[4-(difluoromethoxy)phenyl]methyl}piperidine
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1,2,3-thiadiazole
2-propyl-N-[1-(thian-4-yl)piperidin-4-yl]-1,3-thiazole-4-carboxamide
3-fluoro-N-{1-[1-(oxan-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
5-fluoro-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}quinazolin-4-amine
1-[cyclohexyl(methyl)amino]-3-[2-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-[3-(2-fluorophenoxy)azetidine-1-carbonyl]piperidine-1-carboxamide
(1R,7S)-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-3-(2-methoxyethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-methoxy-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-amino-N-[(5-chloro-1H-indol-2-yl)methyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
N'-cyclopentyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]butanediamide
[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl](pyridin-3-ylmethyl)amine
5-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-hydroxy-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-2-phenylpyrimidine-5-carboxamide
3-[5-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1H-indole
4-[2-(2-fluorophenyl)acetyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
4-methoxy-N-(2-{7-[(8-methoxyquinolin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
3-(3-cyclopentylpropanoyl)-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(4-methyl-1H-imidazole-5-carbonyl)pyrrolidine-2-carboxamide
(3aR,6aR)-2-(cyclopentylcarbamoyl)-5-(1H-imidazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid