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N-cyclopropyl-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-4-(trifluoromethyl)benzamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(1,3-thiazol-2-ylmethyl)-decahydro-2,7-naphthyridine-2-carboxamide
4-(3-chloro-4-methoxybenzoyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
1-(3-methylpiperidin-1-yl)-3-{[3-(morpholin-4-yl)propyl]amino}propan-1-one
N-({8-[(4-methoxy-2,3-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]isoquinoline
3-(5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenol
1-({5-[(4-hydroxyquinolin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
[1-(3-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenyl)ethyl]dimethylamine
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-4,6-dimethoxypyrimidine
7-{[4-(propan-2-yl)phenyl]methyl}-2-(pyrimidin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-[3-(4-fluorophenoxymethyl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
4-{5-[2-(1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1H-indole
1-{3-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}-1H-pyrazole
4-ethyl-2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-5-methylpyrimidine
3-(2-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-2-oxoethyl)-4,6-dimethyl-2,3-dihydro-1H-indol-2-one
6-(cyclopropylmethoxy)-4-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoxaline
3-(1H-1,3-benzodiazol-2-yl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]benzamide
8-(2-aminopyridine-4-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(3-ethoxypropyl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]pyrrolidin-3-yl]-2-(methylamino)acetamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
4-{4-[2-(3-methoxyphenoxy)ethyl]piperazin-1-yl}pyrimidine-5-carboxylic acid
3-{4-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1,3-thiazol-2-yl}pyridine
6-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]-3,4-dihydroquinazolin-4-one
2-[4-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
5-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-8-methoxyquinoline
7-(2-methoxyphenyl)-2-(pyridin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[6-(2,3-dihydro-1-benzofuran-7-yl)pyridin-3-yl]acetic acid
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-amino-6-tert-butyl-4-[5-(hydroxymethyl)furan-2-yl]pyridine-3-carbonitrile
4-[(2,4-difluorophenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-5-(3-phenylpropyl)imidazolidine-2,4-dione
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2-(thiophen-2-yl)acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-phenyl-1,2,4-triazin-3-amine
2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-N-methylpyridine-4-carboxamide
(1S,5R)-6-(3,4-difluorobenzoyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-(1,1-dioxo-1λ6-thian-4-yl)-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
{1-[2-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-1,3-benzodiazol-2-yl}methanol
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
(1R,5S,8R)-N,N-dimethyl-3-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-azabicyclo[3.2.1]octan-8-amine
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-N,N-dimethylpyrimidin-4-amine
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(2-hydroxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-methyl-5-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
2-chloro-5-acetamido-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)benzamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine