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methyl (1R,3S,3aR,6aS)-3-(3-chloro-4-fluorophenyl)-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(3S,4R)-1-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-{4-[4-(azepan-1-yl)piperidin-1-yl]phenyl}-3-methylimidazolidin-2-one
4-(1H-imidazol-1-ylmethyl)-N-[3-(2-oxopyrrolidin-1-yl)phenyl]piperidine-1-carboxamide
N-(2-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
2-methyl-1-phenyl-N-(4H-1,2,4-triazol-4-yl)-1H-1,3-benzodiazole-5-carboxamide
(3R)-1-[5-(methanesulfonylmethyl)pyridin-2-yl]-3,4,4-trimethylpyrrolidin-3-ol
1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-ol
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[(4,4-difluoropiperidin-1-yl)methyl]-2-(3-methylphenyl)pyrimidine
8-(1H-indol-3-ylmethyl)-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-1-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)sulfonyl]-4-(hydroxymethyl)piperidin-3-ol
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
2-(dimethylamino)-N-methyl-N-{2-phenyl-1-[1-(4-phenylbenzoyl)piperidin-4-yl]ethyl}acetamide
1,4,6-trimethyl-3-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
3-acetamido-N-[6-(3-methoxyphenoxy)pyridin-3-yl]pyrrolidine-1-carboxamide
(3aR,5R,6S,7aS)-2-(7,8-dimethylquinolin-4-yl)-octahydro-1H-isoindole-5,6-diol
N-[(3R,4R)-1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(2-fluorophenyl)acetamide
N-ethyl-N-[2-(phenylsulfanyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(2-methylphenyl)-3-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
(3S,4R)-4-(3-fluorophenyl)-1-[2-(3-methoxyphenyl)acetyl]pyrrolidine-3-carboxylic acid
2-({[(3R,4R)-1-(2,3-dimethyl-1H-indole-7-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
3-[(3-fluorophenyl)amino]-N-(2-methoxyphenyl)piperidine-1-carboxamide
3-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-(oxan-4-yl)piperidine
N-[1-(4-cyclopentylpyrimidin-2-yl)pyrrolidin-3-yl]acetamide
2-amino-4-(3-ethoxy-4-hydroxyphenyl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
(2E)-3-(1H-imidazol-4-yl)-1-{4-[5-(3-methoxyphenyl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
methyl (2S)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine-2-carboxylate
{2-oxo-2-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}urea
1-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-(prop-2-en-1-yl)piperidine-3-carboxamide
N-{1-[1-(cyclopropylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-3-(pyrazin-2-yl)propanamide
(1S,5R)-6-(dimethyl-1,2-oxazole-4-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{[3-(furan-2-yl)phenyl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-(dicyclopropylmethyl)-N-methylacetamide
5-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[4-(ethoxycarbonyl)piperazin-1-yl]-2-[2-(methylsulfanyl)phenyl]acetic acid
8-(6-ethyl-2-methylpyrimidin-4-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
6-ethyl-2-methyl-4-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]quinoline
5-[(2,4-dimethoxyphenyl)methyl]-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[(2-benzenesulfonamidopyrimidin-5-yl)methyl]-1-methylpiperazine-2-carboxylic acid
1-(3-chloro-4-methoxyphenyl)-3-(1-methyl-2-oxopyrrolidin-3-yl)urea