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4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{4H-thieno[3,2-b]pyrrol-5-ylmethyl}piperidine
3-(2H-1,3-benzodioxol-5-yl)-5-[2-(propan-2-yloxy)phenoxymethyl]-1,2,4-oxadiazole
2-(pyrrolidin-1-yl)-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-5,6,7,8-tetrahydroquinazoline
2-(4-fluorophenyl)-2-hydroxy-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
(3R,5S)-5-(3-fluorophenoxymethyl)-N-(2-hydroxyethyl)-1-(2-methylpropyl)piperidine-3-carboxamide
{4-[(2-chlorophenyl)methyl]-1-[2-(trifluoromethyl)benzenesulfonyl]piperidin-4-yl}methanol
6-(3-fluorophenyl)-N-methyl-N-(2-phenoxyethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-phenylacetamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-(furan-2-ylmethyl)-3-(1-methyl-1H-pyrazol-5-yl)-N-(pyridin-2-ylmethyl)propanamide
2-fluoro-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-5-sulfamoylbenzamide
methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})(thiophen-3-ylmethyl)amine
4-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]morpholine
N,2-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
3-hydroxy-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-cyclobutyl-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
1-[(2-fluorophenyl)methyl]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-6-oxopiperidine-3-carboxamide
2-[4-(2-ethylbutyl)piperazin-1-yl]-1,3-benzoxazole
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,4-oxazepan-6-ol
[3-(3-phenylpropyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl]methanol
N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylthiophene-3-carboxamide
6-cyclopropyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrimidin-4-amine
4-(3-methylbutyl)-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
N-(2,3-dihydro-1H-inden-2-yl)-1,9-dioxaspiro[5.5]undecan-4-amine
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
6-methoxy-N-{1-[4-(morpholin-4-yl)phenyl]ethyl}pyrimidin-4-amine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-5-methyl-1,3-oxazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-N-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
2-({[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-thiadiazole
3-phenoxy-N-{1-[1-(propane-1-sulfonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
2-[(2S,4S)-2-(diethylcarbamoyl)-4-(4-fluoro-3-methylbenzamido)pyrrolidin-1-yl]acetic acid
{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}({1-[3-(trifluoromethyl)phenyl]propan-2-yl})amine
N-[(2,4-dichloro-6-methylphenyl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-(cyclopropylmethyl)-2-[(2R)-2-hydroxypropanoyl]-N-propyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
3-(4-chlorophenyl)-1-(1,2-oxazolidin-2-yl)-3-phenylpropan-1-one
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
methyl 4-({4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-4-ylmethyl)amino]ethyl]piperidin-1-yl}methyl)benzoate
8-(2-amino-6-methylpyrimidin-4-yl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
2-[(cyclohexylamino)methyl]-4-(pyridin-3-yl)phenol
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
3-(2-ethoxyethyl)-2-oxo-1-(pyrimidin-2-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
(4-methyl-5-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methanol
ethyl 1-(3-fluorophenyl)-5-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1H-pyrazole-4-carboxylate