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4-ethyl-5-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(pyrrolidin-1-yl)benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidine
2-(1H-imidazol-2-yl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]benzamide
dimethyl[(6-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}pyridin-3-yl)methyl]amine
3-(4-benzyl-1H-pyrazol-5-yl)-1-(2-methylfuran-3-carbonyl)piperidine
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S)-2-acetamido-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
ethyl 3-({2-[2-(dimethylamino)ethyl]morpholine-4-carbonyl}amino)propanoate
1-[(3-fluorophenyl)methyl]-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-1,4-diazepane
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)propanamide
1-cyclooctyl-5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2,3,6-trimethylquinoline-4-carboxamide
3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
1,2-dimethyl-4-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine
cyclopentyl 4-({[2-(2-oxoimidazolidin-1-yl)ethyl]carbamoyl}amino)benzoate
3-{[(5,6-dimethylpyrimidin-4-yl)amino]methyl}-2-methoxy-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-[4-chloro-2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyrimidine
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]piperidin-4-amine
2-methyl-6-[2-(pyridin-2-yl)ethyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
4-(1-methylpiperidine-2-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
1-[2-methyl-4-({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
(2R,6S)-4-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-2,6-dimethylmorpholine
3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
1-[9-cyclohexyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(pyridin-3-yloxy)ethan-1-one
2-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]-N,N-dimethyl-2-phenylacetamide
N-[(3S)-1-[3-(piperidin-4-ylmethyl)benzoyl]pyrrolidin-3-yl]acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]-3-methyl-1H-pyrazole-5-carboxamide
2-(4-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}-2-chlorophenoxy)acetamide
2-[2-methyl-4-(4-methylphenyl)-5-oxopiperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
2-{[5-(hydroxymethyl)furan-2-yl]methyl}-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-methyl-1-(naphthalen-1-ylmethyl)-N-(1,2-oxazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-methyl-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]thiophene-2-carboxamide
1-(2-ethylpiperidin-1-yl)-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]ethan-1-one
methyl 2-(ethylsulfamoyl)-6-[4-(trifluoromethyl)benzoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-(3,3-diphenylpiperidine-1-carbonyl)-4-methylpyrimidine
4-(1H-imidazol-1-ylmethyl)-5-methyl-2-(2-methylphenyl)-1,3-oxazole
3-methyl-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-3-phenylbutan-1-one
1-(4-methoxy-3-methylbenzoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
(2S,4S)-4-amino-1-[4-(1H-indol-3-yl)butanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2S,4S)-4-amino-1-[4-(difluoromethoxy)benzenesulfonyl]-N-methylpyrrolidine-2-carboxamide
2-[(4-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-4-(thiophen-2-yl)butanamide
1-methyl-2-(morpholin-4-yl)-N-[(1R)-1-phenylethyl]-1H-1,3-benzodiazole-5-carboxamide