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2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[5-(morpholin-4-yl)pentyl]acetamide
7-[(4-methylphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(3aR,7aS)-N-(1-methyl-1H-indazol-5-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-({4-methyl-5-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
1-(2-fluorophenyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]cyclopropane-1-carboxamide
N-[(3S,4R)-1-(cyclobutylmethyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
N-(3-chloro-4-methoxyphenyl)-6-[(3-methoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-(1H-indazol-7-yl)-1-(oxan-4-yl)urea
2-[2-(methylsulfanyl)phenyl]-N-(propan-2-yl)pyrimidin-4-amine
3-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(6-methoxypyridin-3-yl)urea
N-[3-(5-methyl-4-{[3-(thiophen-2-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]oxane-4-carboxamide
5-methyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-cyclobutyl-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-{3-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]thiophen-2-yl}ethan-1-one
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1-(propan-2-yl)piperidine-3-carboxamide
5-methoxy-N-(2-methoxyethyl)-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-2-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)piperidin-2-one
8-(6-aminopyrimidin-4-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(1-methoxyethyl)-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-hydroxy-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-2-(phenoxymethyl)pyrimidine-5-carboxamide
5-(thiophen-2-yl)-3-[1-(1H-1,2,4-triazol-5-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-amino-4-(5-fluoro-1-methyl-1H-indol-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[(2,6-difluorophenyl)methyl]-N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(2-ethoxypyridin-3-yl)methyl]acetamide
3-(2-fluorophenyl)-5-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-cyclohexyl-5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
1-[4-(pyrimidin-2-yl)piperazin-1-yl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
5-(oxolan-2-yl)-N-[(4-phenyloxan-4-yl)methyl]thiophene-2-carboxamide
methyl[1-(3-methylpyridin-2-yl)propan-2-yl][(1-propyl-1H-imidazol-2-yl)methyl]amine
6-cyano-N-[(3R,4S)-4-(propan-2-yl)-1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]pyridine-3-carboxamide
1-[(4-hydroxyphenyl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
ethyl 4-(3-phenylpropyl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylate
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
2-butyl-8-[(6-methylpyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
7-(5-methyl-1,2-oxazole-3-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[1-(3-phenylpropyl)-5-(1,3-thiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
(1s,4s)-4-[3-(propan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-ol
{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-[(3-methoxyphenyl)methyl]piperidin-4-yl}methanol
N-methyl-2-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
8-[2-(prop-2-en-1-ylsulfanyl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-[2-(pyridin-2-yl)-1H-imidazol-1-yl]-1H-indole
N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2,6,8-trimethylquinoline-4-carboxamide
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(5-methylthiophen-2-yl)methyl]benzamide
3-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,5-dimethyl-1H-pyrazole