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4-fluoro-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
(2R,6R)-4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylacetamide
2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-thiazole-4-carboxamide
7-(2-methoxyethyl)-2-(6-methoxypyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-fluorophenoxy)-1-[4-(methylamino)pyrimidin-2-yl]piperidine-4-carboxylic acid
6-(hydroxymethyl)-N-[4-(1H-pyrazol-5-yl)phenyl]-1,4-oxazepane-4-carboxamide
5-(2-cyclopentylacetamido)-N,1-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
7-(propan-2-yl)-2-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazole
[(1-ethyl-1H-pyrazol-4-yl)methyl][(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]amine
(1S,6R)-9-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
5-(3-fluorophenoxymethyl)-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
1-(4-ethyl-5-methylpyrimidin-2-yl)-4-(hydroxymethyl)azepan-4-ol
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[methyl(propan-2-yl)amino]pyridine-3-carboxamide
4-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
N-(furan-2-ylmethyl)-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[(2-chlorophenyl)methyl]-4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
(2S)-N-(2-ethyl-1H-1,3-benzodiazol-6-yl)-2-(piperidine-1-carbonyl)pyrrolidine-1-carboxamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
1-[(3-fluoro-4-methoxyphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
4-methyl-2-(2-oxo-2-{4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethyl)-1,2-dihydrophthalazin-1-one
2-chloro-4-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenol
1-[1-(3-phenylpropyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
N-[2-(dimethylamino)ethyl]-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-N-methylpiperidin-3-amine
1-(2-fluorophenyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}cyclopropane-1-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylfuran-2-carboxamide
4-[(dimethylamino)methyl]-1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]azepan-4-ol
N-(3-chloro-4-methoxyphenyl)-4-(pyridin-4-yl)piperidine-1-carboxamide
2-[(benzyloxy)methyl]-5,6-dimethyl-1H-1,3-benzodiazole
2-benzyl-8-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decan-3-one
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
ethyl 2-amino-4-(2-butyl-1H-imidazol-4-yl)-3-cyano-5,6,7,8-tetrahydro-1,6-naphthyridine-6-carboxylate
5-(propan-2-yl)-3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2-oxazole
N-cycloheptyl-3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propanamide
2-{5-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-phenyl-1,2-oxazole-5-carboxamide
3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-[2-(piperidin-1-ylmethyl)phenyl]urea
3-{1-[(3-chloro-1-benzothiophen-2-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
N-butyl-3-({[3-(1H-indol-1-yl)propyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-2-(methoxymethyl)-6-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
4-(1-benzyl-1H-pyrazol-4-yl)-1-[2-(1H-pyrrol-1-yl)ethyl]-1,2,3,6-tetrahydropyridine
4-(3,4-difluorobenzoyl)-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
5-{[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]methyl}thiophene-2-carboxylic acid
2-methoxy-4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1,3-thiazole-5-carboxamide
(3S,4S)-1-[(2-ethylpyrimidin-4-yl)methyl]-4-(3-methoxyphenyl)piperidin-3-ol
4,4-difluoro-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidine
4-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-oxaspiro[4.4]nonan-2-one