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1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-(ethylsulfanyl)propan-1-one
1-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-ethyl-3-(4-hydroxyphenyl)-N-(oxolan-2-ylmethyl)propanamide
3-[({1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
2-(4-chlorophenyl)-1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazole
4-[(4-fluorophenyl)methyl]-1-[2-(1H-imidazol-1-yl)ethyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-[({pyrazolo[1,5-a]pyridin-3-ylmethyl}amino)methyl]piperidin-3-ol
4-({4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(methoxymethyl)piperidine
{1-[3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]cyclopropyl}methanol
N-(3-{4-[(oxan-4-yl)amino]piperidin-1-yl}phenyl)-3-(trifluoromethyl)benzamide
N-cyclopropyl-5-[2-(1H-indazol-1-yl)acetyl]-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(1-ethyl-1H-pyrazol-4-yl)-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methylquinoline-4-carboxamide
2-[4-(2-methyloxane-2-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
N-(4-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenyl)acetamide
1-cyclohexyl-3-cyclopropyl-5-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazole
2-methyl-8-(quinoxaline-5-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(5-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)-1H-1,3-benzodiazole
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
8-[(2E)-hex-2-en-1-yl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{3-[3-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
4-[(furan-2-ylmethyl)amino]-N-(1-methoxybutan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-3-(2-methoxyphenyl)-N-[(3S)-2-oxoazepan-3-yl]propanamide
2-{2-[1-(1-benzothiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
7-(cyclopropylmethyl)-2-(2,3-dihydro-1H-inden-2-yl)-2,7-diazaspiro[4.5]decan-6-one
7-(3-chlorophenyl)-4-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}azepan-4-amine
5-{1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({methyl[2-(methylamino)ethyl]amino}methyl)piperidin-2-one
N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(2-phenylethyl)acetamide
1-[4-(1H-pyrazol-3-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-(2-hydroxyethyl)-5-methoxy-3-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
N-(4-{[4-(4-benzyl-2,5-dioxoimidazolidin-4-yl)piperidin-1-yl]methyl}phenyl)acetamide
dimethyl(2-{2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
(1S,5R)-3-{[3-(benzyloxy)-4-methoxyphenyl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-1-{2-[1-(3,5-dimethoxybenzoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
4-(benzyloxy)-1-(3,5-difluorobenzoyl)piperidine
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-3-(1-methylcyclohexanecarbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(4-fluorophenyl)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-amine
(3S,5R)-5-(cyclopropylcarbamoyl)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine-3-carboxylic acid
(3aR,6aR)-2-(2-cyclopentylacetyl)-5-(3-methoxypropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(4-ethyl-1,3-thiazol-2-yl)methyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
5-(2,6-difluoro-4-methoxyphenyl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzothiophene-2-carboxamide
methyl 4-[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)carbamoyl]butanoate
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
(4aS,8aR)-1-(2-aminoethyl)-6-[1-(4-methylphenyl)cyclopropanecarbonyl]-decahydro-1,6-naphthyridin-2-one
4-(1-{5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyrimidine