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ethyl 4-[(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
1-(2-ethoxyethyl)-3-[2-(2-fluorophenyl)ethyl]piperidine
3-(2-phenylethyl)-7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(4aS,7aR)-1-benzoyl-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
dimethyl[(5-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}thiophen-3-yl)methyl]amine
1-[4-(2-oxopyrrolidin-1-yl)butanoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-amine
5-(3-fluoro-4-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(adamantan-1-ylmethyl)-7-fluoro-N-(2-hydroxyethyl)-3-methyl-1-benzofuran-2-carboxamide
(4aS,7aR)-N-[2-(4-fluorophenyl)ethyl]-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
N-(2-methylpropyl)-2-(morpholin-4-yl)-N-(thiophen-3-ylmethyl)pyridine-3-carboxamide
(3S,5R)-5-(cyclopropylcarbamoyl)-1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-3-carboxylic acid
5-(2-methylpropyl)-1'-(5-propyl-1,3,4-thiadiazol-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(4-{2-[4-(furan-3-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
N-(2-{[7-acetyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethyl)acetamide
N-[1-(2-phenylethyl)piperidin-3-yl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-amino-4-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
3-[2-(methylsulfanyl)benzoyl]-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine
3-chloro-4-({1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}oxy)-N-[2-(dimethylamino)ethyl]benzamide
4-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-benzoyl-N-(1-benzothiophen-5-ylmethyl)piperidin-4-amine
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-ethyl-N-[(5-methylfuran-2-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
3-(4-methylpiperazine-1-carbonyl)-1-propyl-N-{[3-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{1-[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
3-[1-benzyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiolane-1,1-dione
[(2-ethylpyrimidin-5-yl)methyl]({[2-(2-fluorophenoxy)pyridin-3-yl]methyl})amine
1-[2-(4-butyl-2,3-dioxopiperazin-1-yl)-2-phenylacetyl]piperidine-4-carboxamide
6-ethyl-3-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,5-dimethyl-1,2-dihydropyridin-2-one
1-{[4-(6-chloropyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}cyclopentane-1-carboxylic acid
2-{5-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrole-2-carbonyl]-1H-pyrazol-3-yl}phenol
2-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(3-hydroxy-3-methylbutyl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]benzamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide
N-{3-[3-(azocan-1-ylmethyl)phenoxy]propyl}-3-(2-oxoimidazolidin-1-yl)benzamide
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}(methyl)[3-(1H-pyrazol-1-yl)propyl]amine
6-fluoro-3-(morpholin-2-ylmethyl)-3,4-dihydroquinazolin-4-one
1-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
1-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
4-chloro-1-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2-[2-(dimethylamino)ethyl]-9-[(2-fluoro-5-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-butyl-4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,2-diethylcyclopropane-1-carboxamide
methyl({[3-({1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}methoxy)phenyl]methyl})(quinolin-6-ylmethyl)amine
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
5-{2-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one