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(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
4-({2-[1-(thiophene-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-methyl-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-hydroxy-3-[(4-methylpiperidin-1-yl)methyl]-1-(3-phenylpropyl)piperidin-2-one
9-methoxy-7-(6-methoxypyridin-2-yl)-4-{[4-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{methyl[2-(pyridin-4-yl)ethyl]sulfamoyl}-N-(prop-2-en-1-yl)benzamide
7-[1-(4-methoxyphenyl)piperidin-4-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(4-methylpyridin-2-yl)methyl]acetamide
(1R,5R)-N,N-dimethyl-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methylazepane-2-carboxamide
1-[cyclohexyl(methyl)amino]-3-[3-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-(2,3-dihydro-1H-inden-2-yl)-3-(3,4-dimethoxybenzoyl)piperidine
6-methyl-2-oxo-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-1,2-dihydropyridine-3-carboxamide
3-(2,2,6,6-tetramethylpiperidin-4-yl)-3,4-dihydroquinazolin-4-one
2,6-dimethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]quinoline-4-carboxamide
4-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-[3-(pyridin-2-yl)azetidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
{3-[(2-methylphenyl)methyl]-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperidin-3-yl}methanol
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl){[1-(propan-2-yl)piperidin-3-yl]methyl}amine
2-[(2-cyclohexylpyrimidin-5-yl)methyl]-7-ethyl-2,7-diazaspiro[4.5]decan-6-one
2-methyl-5-({4-[3-(piperidin-1-yl)azetidine-1-carbonyl]piperidin-4-yl}oxy)pyridine
{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amine
N-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-1-(pyridin-2-ylmethyl)piperidin-4-amine
(3aR,6aR)-N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(2S,4S)-1-[(4-phenylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
2-[4-(1H-indol-3-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
1-{1-[(3-chloro-2,6-difluorophenyl)methyl]piperidin-4-yl}piperidin-4-ol
(1S,5R)-6-(2-methoxyethyl)-3-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(2-fluorophenyl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]-3-phenylpropanamide
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(2-methoxyethyl)(propan-2-yl)amine
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(morpholin-2-yl)acetamide
5-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(2-fluoro-3-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(1,4-oxazepane-4-sulfonyl)-N-[(3S)-pyrrolidin-3-yl]benzamide
1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-[3-({[3-(2-hydroxyphenyl)propyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
5-ethyl-2-(1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)pyridine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
N-(butan-2-yl)-N-[(4-chlorophenyl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
methyl 4-[4-(8-methoxyquinolin-2-yl)piperazin-1-yl]benzoate
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-butyl-3-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(dimethyl-1,2-oxazol-4-yl)-4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
6-[1-(3,3-dimethylcyclohexyl)piperidin-4-yl]-2-[2-(pyridin-2-yl)ethyl]-3,4-dihydropyrimidin-4-one
3-methyl-7-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-[5-(methanesulfonylmethyl)pyridin-2-yl]phenol
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(pyridine-2-carbonyl)piperazine