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3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(2-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-benzyl-5-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-4-yl)imidazolidine-2,4-dione
2-[1-(2-phenylethyl)-4-(9H-purin-6-yl)piperazin-2-yl]ethan-1-ol
4-({1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}methyl)-1-phenyl-1H-1,2,3-triazole
4-benzyl-2-{[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}morpholine
1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-(4-methoxyphenoxy)piperidine
2-methoxy-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-5,6,7,8-tetrahydroquinazolin-2-amine
(2R)-2-{[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-3-phenylpropan-1-ol
N-(4-methoxy-2-methylphenyl)-3-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]propanamide
N-(furan-2-ylmethyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carboxamide
2-[(3,3-diphenylpiperidin-1-yl)methyl]pyrimidine
(1R,2R,6S,7S)-4-[4-(5-methylfuran-2-yl)benzoyl]-4-azatricyclo[5.2.1.02,6]decane
2-methoxy-4-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
3-(3-methyl-1,2-oxazol-5-yl)-4-pentyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(7-{[5-(3-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclopropanecarboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1,3-dimethyl-1H-pyrazole-4-carboxamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)(propan-2-yl)amine
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-[2-(trifluoromethyl)phenyl]acetamide
N-(3,4-difluorophenyl)-1-(5-methyl-1H-indazole-3-carbonyl)piperidin-3-amine
3-ethoxy-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
(7S,8aS)-2-methyl-7-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[cyclopentyl(methyl)amino]-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
1-[(3-fluorophenyl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-2-yl)propan-1-one
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-(naphthalen-2-ylmethyl)piperazin-2-one
methyl 3-[(3S,4R)-1-[(3-methoxyphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
N-(1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-yl)acetamide
7-cyclopentyl-2-(1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-(4-methylpiperidine-1-carbonyl)-4-oxo-N-(2-phenylethyl)-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
(2R,6R)-4-(2-hydroxy-4-methoxybenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N'-(3-ethylphenyl)-N-[(5-methylpyrazin-2-yl)methyl]butanediamide
N-methyl-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-[1-(naphthalen-2-yl)ethyl]acetamide
1-[(3,3-dimethyl-4-phenylpyrrolidin-1-yl)sulfonyl]-4-methoxypiperidine
8-(1,3-benzoxazol-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]pyridin-3-ol
N-cyclopentyl-5-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-cyclopropyl-5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,2,4-triazole
N-[(3S,4R)-1-(3-chloropyridin-2-yl)-4-propylpyrrolidin-3-yl]acetamide
3-(2-fluoro-5-methoxyphenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
propyl 4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
4-[(2,3-difluorophenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-(1-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
N-{2-[3-(propan-2-yloxy)phenyl]ethyl}-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide