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{2-[(2-ethyl-6-methylpyrimidin-4-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
(1S,4S)-2-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]-2-azabicyclo[2.2.1]heptane
(3S,4S)-N-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-hydroxy-4-(morpholin-4-yl)pyrrolidine-1-carboxamide
2-(2-methoxyethyl)-9-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-{5-[3-(4-chlorophenyl)propyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2,2,2-trifluoroethyl)acetamide
N-[(3R)-piperidin-3-yl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-methyl-N-({3-[(1-methylpiperidin-4-yl)methyl]-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl}methyl)aniline
2-{5-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
3-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzene-1-sulfonamide
1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-(pentan-2-yl)-4-phenyl-1H-imidazole
2-methoxy-5-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}pyridine
N-[2-(4-fluorophenoxy)ethyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-(2-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-(propan-2-yl)piperidine-4-carboxamide
methyl 2-{4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
[4-(2-phenoxyethyl)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-4-yl]methanol
N-cyclopropyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-(2-methoxyethyl)-4-methyl-3-{[(5-methylpyridin-3-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
6-({[1-(ethoxymethyl)cyclobutyl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-(2,1,3-benzothiadiazol-4-yl)-3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
N-[2-(3-methoxy-4-propoxyphenyl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
[(2Z)-2-chloro-3-phenylprop-2-en-1-yl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-(4-fluorophenyl)-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-3-amine
methyl 2-[1-(2-methoxypyridine-4-carbonyl)-3-oxopiperazin-2-yl]acetate
(4aS,7aR)-1-(3,5-dimethylbenzenesulfonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-{[1-(1-cycloheptylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
(2S,4S)-4-amino-1-[(2-cyclohexylpyrimidin-5-yl)methyl]pyrrolidine-2-carboxylic acid
2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-N-(cyclohexylmethyl)acetamide
4-hydroxy-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-cyclopropyl-2-[1-(2-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
1-[(1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-(cyclopropylmethyl)-2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3S,4S)-1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(piperidin-1-yl)pyrrolidin-3-ol
2-(2,4-dichlorophenoxy)-N-[1-(1,3-thiazol-5-yl)propan-2-yl]acetamide
N-{1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]pyrrolidin-3-yl}acetamide
N-butyl-1-(cyclohexylmethyl)-6-oxopiperidine-3-carboxamide
N-{1-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]-1H-pyrazol-4-yl}thiophene-3-carboxamide
1-(2-chloro-4-fluorobenzoyl)-4-(hydroxymethyl)azepan-4-ol
(2S)-2-amino-1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-3-(1H-imidazol-4-yl)propan-1-one
5-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
[1-({[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)cyclobutyl]methanol
(1R,5S,8R)-8-methoxy-3-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3-azabicyclo[3.2.1]octane
2-(1H-pyrazol-1-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}butanamide
3-(4-hydroxyphenyl)-N-(1,2-oxazol-3-ylmethyl)-2-phenylpropanamide
{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(3-phenylpropyl)piperidin-3-yl}methanol
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)propanamide
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one