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N-{2-methoxy-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propanamido]phenyl}benzamide
1-[(3-methoxyphenyl)methyl]-N-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-3-amine
7-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-[2-(1H-imidazol-1-yl)ethyl]-3-[(2-methylbutyl)amino]-5-(pyrrolidine-1-sulfonyl)benzamide
3-methoxy-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide
N-cyclopentyl-3-{methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfamoyl}benzamide
8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
2-{4-[(4-acetyl-1,4-diazepan-1-yl)methyl]phenyl}-6-(2-methoxyethyl)-3,4-dihydropyrimidin-4-one
2-{[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl}pyrimidine
1-methyl-9-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
3-{[4-(trifluoromethoxy)phenyl]methyl}-1,3-oxazolidin-2-one
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-(3-phenoxypropyl)-1H-1,3-benzodiazole-5-carboxamide
6-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,2-dimethylquinoline-4-carboxamide
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(3-methylthiophen-2-yl)formamido]acetic acid
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}propane-2-sulfonamide
3-(4-fluorophenoxymethyl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
8-(6-methoxypyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{2-[1-(4,6-dimethylpyridine-3-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
5-(3,5-difluoropyridine-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-methoxy-1-{1'-[3-(methylsulfanyl)butyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
6-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-N,N-dimethylpyrazine-2-carboxamide
(3aS,6aR)-5-[(5-methylthiophen-2-yl)methyl]-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-(ethylsulfanyl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]propan-1-one
2-[4-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
4-({ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-benzyl-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3-chloro-4-methoxyphenyl)-3-{1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}propanamide
N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
N-benzyl-3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-N-methylpropanamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-fluoro-2-methylbenzamide
N-{2-[methyl(phenyl)amino]propyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-(dimethylamino)-N-methyl-N-(2-phenyl-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}ethyl)acetamide
3-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
4-[5-(3-phenyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridine
4-[2-(1H-pyrazol-1-yl)benzoyl]-1λ6-thiomorpholine-1,1-dione
dipropyl({4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)amine
N-(4-chlorophenyl)-4-[5-(2-methylbenzamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
7-(3-phenylpropyl)-2-(quinoline-3-carbonyl)-2,7-diazaspiro[4.5]decane
(3aR,6aR)-2-cyclopentyl-5-[(6-ethoxypyridin-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-benzyl-4-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperazin-2-one
2-methyl-6-{pyrazolo[1,5-a]pyridin-7-yl}pyridine-4-carboxylic acid
(3R,4R)-1-[(2-methyl-1H-indol-3-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-(oxolan-3-yl)benzamide
(1H-1,3-benzodiazol-2-ylmethyl)({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-methyl-5-{2-oxo-2-[3-(3-phenylpropanoyl)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(4-methoxyphenyl)methyl]acetamide