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N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-7-oxo-3-[2-(thiophen-3-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
3-{1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-1-methyl-1H-imidazole-4-sulfonamide
dimethyl({2-[1-(2-methylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl})amine
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-methyl-1,3-thiazole-4-carboxamide
3-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}azetidin-3-yl)pyridine
5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methyl-2-(pyridin-3-yl)pyrimidine
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-(1,3-thiazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]pyrrolidine-1-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(morpholin-3-yl)acetamide
{1-[4-(1H-pyrazol-5-yl)benzoyl]piperidin-4-yl}(pyridin-2-yl)methanol
7-[(3,4-difluorophenyl)methyl]-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
1-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
2-cyclopropyl-4-methyl-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)pyrimidine-5-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyridin-4-yl)piperazine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
2-methyl-6-{3-[2-(methylsulfanyl)ethyl]-5-[(pyridin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}pyridine
(1S,5R)-6-methyl-3-{[3-(5-methylfuran-2-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{5-[({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}carbamoyl)amino]-2-methoxyphenyl}propanamide
(1R,3S)-N3-ethyl-N1-(1H-indol-4-ylmethyl)-1,2,2-trimethylcyclopentane-1,3-dicarboxamide
N,2-dimethyl-6-(piperidin-4-yl)-N-(quinolin-8-ylmethyl)pyrimidin-4-amine
(3S,9aR)-3-(4-aminobutyl)-8-(3,5-dichlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-(2-phenylethyl)-2-(quinoline-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
[1-(2-amino-6-methylpyrimidin-4-yl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
2-(1-methyl-3-oxopiperazin-2-yl)-N-[2-(propan-2-yloxy)ethyl]acetamide
6-ethyl-4-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
3-[(1,2-oxazol-3-ylmethyl)sulfamoyl]-N-[2-(pyridin-4-yl)ethyl]benzamide
4-(5-chloro-2-methylphenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{[benzyl(methyl)amino]methyl}-N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-phenylpyrrolidin-3-yl]-3-methanesulfonylpropanamide
N-[1-(3-methylpyridin-2-yl)ethyl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
4-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-(cyclohexylmethyl)-4-(pyridin-3-ylmethyl)morpholine
N-{4-[({[2-(butan-2-yloxy)phenyl]methyl}carbamoyl)methoxy]phenyl}propanamide
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-(methylamino)acetamide
[3-benzyl-1-(6-phenylpyridazin-3-yl)piperidin-3-yl]methanol
N-(3-acetamido-4-fluorophenyl)-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
3-methyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-methyl-4-propyl-6-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidine
2-[4-(6-aminopyridine-3-carbonyl)-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
3-chloro-5-fluoro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
(1S,5R)-3-(8-chloroquinoline-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl})amine