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1-[1-(2-cyclopropyl-1,3-benzoxazole-6-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
3-fluoro-N-({7-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
3-{[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(1-methanesulfonylpiperidin-4-yl)urea
8-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-(4-fluorophenyl)-1-(pyrrolidine-1-carbonyl)piperidine
3-phenyl-1-(1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-3-yl)propan-1-one
N-{[1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)piperidin-3-yl]methyl}furan-2-carboxamide
1-{2-[4-phenyl-5-(thiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
N-[(1-benzylpiperidin-4-yl)methyl]-N-methylpyrazin-2-amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(pyridin-2-ylmethyl)amino]pyridine-3-carboxamide
3-(5-methylfuran-2-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
1-[(4-methoxyphenyl)methyl]-N-methyl-N-(1H-pyrazol-5-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-ethyl-N,4-diphenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(quinazolin-4-yloxy)acetamide
2-(cyclopropylmethyl)-7-{2,8-diazaspiro[4.5]decane-3-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
2-[1-(2,2-dimethylpropyl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]oxane-4-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-[4-(morpholin-4-yl)butan-2-yl]-1-(3-phenoxyphenyl)urea
3-[(3R,4S)-4-(dimethylamino)-1-(2-oxo-2-phenylacetyl)piperidin-3-yl]propanoic acid
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-(morpholin-4-yl)butan-1-one
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{[2-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)phenyl]methyl}-1H-pyrazole
1-[2-(methylsulfanyl)ethyl]-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
1-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(3,5-dimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-({5-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
N-methyl-N-[2-(oxan-2-yl)ethyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
3-benzyl-7-[4-(2,5-dimethoxybenzoyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-4-(pyridin-3-ylmethyl)piperazin-2-yl}ethan-1-ol
4-({5-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-methyl-N-[3-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]propanamide
1-(ethanesulfonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
3-(3-chlorophenyl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-3-(pyrrolidin-1-ylmethyl)-1,2,4-oxadiazole
1-[(4-fluorophenyl)methyl]-4-[(1-methyl-1H-indol-6-yl)methyl]piperazin-2-one
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(1-methylcyclopropyl)propan-1-one
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
3-({[1-(2-phenylbenzoyl)piperidin-3-yl]oxy}methyl)pyridine
methyl 3-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-2-propyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-4-carboxamide
2-{[2-(3-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-4-methoxyphenol
N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-N-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide