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7-fluoro-N,N-dimethyl-2-[1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
5-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
2-[4-(2,6-diaminopyrimidin-4-yl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
methyl 4-(5-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
methyl 1-methoxy-2-oxo-8-[2-(thiophen-3-yl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
1-(2-aminoethyl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
4-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-4-oxobutane-1-sulfonamide
(3aR,6aR)-2-cyclopropanecarbonyl-N-[(2,3-difluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4,6-dimethylpyrimidine
N-cyclopentyl-1-ethyl-3-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrazole-5-carboxamide
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-4-(1H-imidazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
2-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
6-chloro-2-methyl-N-[3-(4-methylpiperazin-1-yl)butyl]imidazo[1,2-a]pyridine-3-carboxamide
2-(2-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
(1R,2R)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2-phenylcyclopropane-1-carboxamide
9-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N-[(3S,5S)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
5-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]-4-ethyl-1,3-thiazol-2-amine
5-(3-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
4-{5-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]furan-2-yl}-2-methylbut-3-yn-2-ol
2,8-dimethyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}quinoline-4-carboxamide
(furan-3-ylmethyl)(methyl){[3-({1-[4-(morpholin-4-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
(1-{1-[(5-ethylthiophen-2-yl)sulfonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-methoxy-4-[4-(1H-pyrazol-1-yl)butan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(4-fluorophenyl)-5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
2-(morpholin-4-yl)-6-[2-(morpholin-4-ylmethyl)phenyl]pyrimidin-4-amine
1-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}imidazolidin-2-one
1-ethyl-4,6-dimethyl-3-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-6-(2-methoxyphenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
N-(2,4-dimethoxyphenyl)-3-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]propanamide
(3aR,6aR)-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-{1-[(1S)-2-hydroxy-1-phenylethyl]-4-phenyl-1H-imidazol-5-yl}-2-methoxyphenol
4-[4-(morpholine-4-carbonyl)pyridin-2-yl]-2-(trifluoromethyl)morpholine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(2,5-dimethoxyphenyl)-N-methylacetamide
3-methanesulfonyl-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]propanamide
3-[4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
1-[2-(1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
4-benzyl-3-[1-(4-hydroxybenzoyl)piperidin-4-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-(4-fluoro-3-methoxybenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-({pyrazolo[1,5-a]pyridin-3-ylmethyl}amino)-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
2-[4-(2-chloro-5-methylphenyl)-1H-pyrazol-1-yl]propanamide
N-[2-(dimethylamino)-3-methylbutyl]-6-(propan-2-yl)pyrimidin-4-amine
N-[2-(7-{[4-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-1-methylpiperidine-3-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-propanamidobenzamide
3-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one