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5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-methyl-N-(pyridin-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
1-ethyl-4-({2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1H-pyrrole-2-carbonitrile
N-{1-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-1H-pyrazol-4-yl}-3-phenoxypropanamide
2-methyl-4-{3-[4-(3-methylpyridin-4-yl)piperazine-1-carbonyl]phenyl}butan-2-ol
5-{methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
6-methyl-2-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-N-[(4-methylphenyl)methyl]propanamide
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
2-(oxolan-2-ylmethyl)-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
N-[(4-methoxypyridin-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-fluoro-N-[4-(4-{[2-(4-methoxyphenyl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[4-(dimethylamino)phenyl]ethan-1-one
1-(2-chloro-4-fluorophenyl)-3-[(1R,2S)-2-(methoxymethyl)cyclopentyl]urea
2-(2-aminoethyl)-N-[2-(2,3-dimethoxyphenyl)ethyl]quinazolin-4-amine
2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-5-propyl-1,3,4-oxadiazole
(2-methoxyethyl)({[3-(3-methoxyphenyl)oxolan-3-yl]methyl})[(3-methylthiophen-2-yl)methyl]amine
8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-[2-(thiophen-2-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
3-[5-(pyrazin-2-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(3-methoxypropyl)-1H-pyrazole-4-carboxamide
3-[2-(morpholin-4-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-[3-(4-methoxypiperidine-1-carbonyl)benzenesulfonyl]-4-methyl-1,2,3,6-tetrahydropyridine
(2R)-2-amino-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-methoxypropan-1-one
N-cyclopentyl-N-[2-(dimethylamino)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-(1-hydroxy-2-methylpropan-2-yl)-1-(4-methoxyphenyl)-2,2-dimethylcyclopropane-1-carboxamide
7-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-[4-(3-hydroxynaphthalene-2-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
2-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-8-azabicyclo[3.2.1]octane
N-{2-[4-(2,3-dihydro-1H-inden-2-yl)morpholin-2-yl]ethyl}cyclobutanecarboxamide
methyl 6-[(2E)-4-methylpent-2-enoyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methyl-1-oxobutan-2-yl}acetamide
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-2-(1,2-oxazolidin-2-yl)pyridine
1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S)-1-acetyl-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-methyl-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl](quinolin-8-ylmethyl)amine
N-benzyl-3-(2-{[(5-methylfuran-2-yl)methyl]carbamoyl}ethyl)piperidine-1-carboxamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]pyridine-4-carboxamide
N-[3-({[(3-ethoxy-2-hydroxyphenyl)methyl]amino}methyl)-5-(piperidine-1-carbonyl)phenyl]methanesulfonamide
1-methyl-2,4-dioxo-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
N-(4-tert-butylphenyl)-4-(pyridin-2-ylmethoxy)piperidine-1-carboxamide
4-(1H-imidazol-2-yl)-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole
N-ethyl-4-(2-methoxyphenyl)-6-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
6-methyl-5-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-2-oxo-1,2-dihydropyridine-3-carbonitrile
3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazol-5-amine
3,6-dimethyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-benzofuran-2-carboxamide