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N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-(quinazolin-4-yloxy)acetamide
[(dimethyl-1,2-oxazol-4-yl)methyl]({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl})methylamine
4-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-N-(propan-2-yl)-1,3-oxazole-5-carboxamide
1-(4-{[4-(1-methylazepane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
1-ethyl-8-{[1-(propan-2-yl)-1,2,3,4-tetrahydroquinolin-6-yl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-cyano-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyridine-3-carboxamide
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
N4-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-[(3-chlorophenyl)methyl]-3-[1-(oxolane-3-carbonyl)piperidin-4-yl]propanamide
4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-N-[2-(pyridin-3-yl)ethyl]pyridin-2-amine
N-methyl-2,6-dioxo-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-({7-[2-(3-chlorophenoxy)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-methylthiophene-2-carboxamide
2-[(3,4-dimethoxyphenyl)methyl]-N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
3-({1-[2-(2-methoxyphenoxy)ethyl]piperidin-3-yl}methyl)pyridine
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(benzyloxy)phenyl]-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]ethan-1-one
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(methylsulfanyl)ethan-1-one
4-[(5,6,7-trimethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1λ6-thiomorpholine-1,1-dione
3-(3-hydroxy-1,2-oxazol-5-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
4-cyclopentyl-N-[(4-methanesulfonylmorpholin-2-yl)methyl]pyrimidin-2-amine
1-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethan-1-ol
(3S,9aR)-8-(2-phenylethyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(4-ethyl-5-methylpyrimidin-2-yl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(1-{7-[(3-ethoxy-4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
2-(4-ethoxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
methyl 4-(methylsulfanyl)-2-[3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamido]butanoate
N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-pyrazole-4-carboxamide
5-(azepane-1-carbonyl)-N-[(2-methoxynaphthalen-1-yl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
{1-[5-(cyclooctylamino)-5,6,7,8-tetrahydroquinazolin-2-yl]piperidin-4-yl}methanol
methyl 1-(naphthalen-2-ylmethoxy)-2-oxo-8-(quinolin-7-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-{4-[7,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
2-[(5-methylpyrazin-2-yl)methyl]-9-(pent-4-enoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(cyclopropylmethyl)-7-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(2-methanesulfonylethyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
methyl (2S)-2-amino-5-[4-(2-methoxybenzoyl)piperazin-1-yl]-5-oxopentanoate
(benzylsulfamoyl)[2-(pyridin-2-ylsulfanyl)ethyl]amine
N-[(5-methylpyrazin-2-yl)methyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
(4aS,8aR)-6-(2,3-dihydro-1H-indene-5-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
6-[(3-aminopyrrolidin-1-yl)methyl]-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-4-(1H-pyrazol-1-yl)benzamide
[(1S)-1-[1-(cyclohexylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl](methyl)amine