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4-(1H-imidazol-1-ylmethyl)-1-(2,3,6-trimethylquinoline-4-carbonyl)piperidin-4-ol
N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2H-1,3-benzodioxole-5-carboxamide
1-ethyl-5-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]piperidin-2-one
5-fluoro-3-methyl-2-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1H-indole
methyl 3-chloro-4-({[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]carbamoyl}amino)benzoate
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-2-one
N-({7-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-[1-(pyrazin-2-yl)piperidin-3-yl]acetamide
2-(4-{[3-({1-[(E)-2-phenylethenesulfonyl]piperidin-4-yl}oxy)phenyl]methyl}piperazin-1-yl)pyrimidine
4-[2-(pyridin-3-yl)morpholine-4-carbonyl]benzene-1-sulfonamide
N-[2-(2-chloro-6-fluorophenyl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)piperidin-3-ol
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
3-{1-[(5-chlorothiophen-2-yl)sulfonyl]piperidin-4-yl}-N-phenylpropanamide
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-methanesulfonylethan-1-one
5-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
3-(3,4-dimethoxybenzoyl)-N-ethylpiperidine-1-carboxamide
1-(3,5-dimethylfuran-2-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(methylsulfamoyl)ethyl]acetamide
2-hydroxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
N-[(2-ethoxyphenyl)methyl]-N-ethyl-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}piperidine-1-sulfonamide
2-{1-cyclohexyl-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
5-acetyl-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}thiophene-2-carboxamide
ethyl 2-{1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}acetate
5-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]pyridine-2-carbonitrile
N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)-2-methylpyridine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]benzamide
3-(azocan-1-yl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methylpropanamide
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxo-N-phenylacetamide
N4-methyl-N2-{1-oxaspiro[4.4]nonan-3-yl}pyrimidine-2,4-diamine
3-[2-({[(4,6-dimethylpyridin-3-yl)methyl]carbamoyl}amino)phenyl]-N-methylpropanamide
(4S)-4-acetamido-4-[1-methyl-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]butanamide
4-(4-chlorophenyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}butanamide
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-4-(1H-pyrazol-3-yl)benzamide
1-(2-ethoxyethyl)-5-(3-hydroxyazetidine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]pyrazin-2-ol
3-[1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydroquinoxalin-2-one
6-(difluoromethyl)-2-[4-({[(3-methoxyphenyl)methyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
1-ethyl-4-{[methyl({2-methylthieno[2,3-d]pyrimidin-4-yl})amino]methyl}pyrrolidin-2-one
4-(1H-pyrazol-3-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
2-(4-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
3-{2-[2-(3-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-[1-({3-[3-(morpholin-4-yl)propoxy]phenyl}methyl)azetidin-3-yl]morpholine
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide