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8-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[(2-fluorophenyl)methyl]-11-{[2-(pyridin-2-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
[(2R)-1-[8-chloro-2-(furan-2-yl)quinoline-4-carbonyl]pyrrolidin-2-yl]methanol
[5-({3-[(4-methoxyphenyl)amino]piperidin-1-yl}methyl)furan-2-yl]methanol
6-[1-(3-chloro-2-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-{4-[methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]piperidin-1-yl}ethan-1-one
5-[4-fluoro-3-(hydroxymethyl)phenyl]pyridin-2-ol
methyl 2-{[(4-fluorophenyl)methyl]sulfamoyl}-6-(thian-4-yl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3S,4R)-4-propyl-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanesulfonamide
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-2-(4-methoxypiperidin-1-yl)pyridine
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
3-[(4-benzoylpiperazin-1-yl)methyl]-4-chloro-1-methyl-1H-indazole
6-(methoxymethyl)-1-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,5R)-6-benzyl-3-(furan-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3aS,6aS)-2-[3-(4-chlorophenyl)propanoyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[3-benzyl-1-(2-chlorophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclopropylacetamide
2-[1-(5-chloro-2-methoxyphenyl)-5-[1-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
(3S,4S)-1-(5-fluoro-1H-indole-2-carbonyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
methyl 2-{4-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
N-{4-[5-methyl-4-({spiro[2.5]octan-1-ylformamido}methyl)-1,3-oxazol-2-yl]phenyl}furan-3-carboxamide
4-[2-(dimethylamino)ethyl]-11-{[(1-phenylcyclohexyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(thiolan-3-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)methyl]thiophene-2-sulfonamide
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyethoxy)piperidine
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)-1H-indole-5-carboxamide
(1S,5R)-3-benzoyl-N-[(4-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
4-{1-[1-(5-chloro-2-fluorobenzoyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-(oxolan-2-ylmethyl)-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-{[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
1-{4-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
methyl 2-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]pyridine-3-carboxylate
5-acetyl-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]thiophene-3-carboxamide
1-methyl-9-(prop-2-en-1-yl)-4-(pyrrolidine-1-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
3-[3-(oxan-4-yl)-5-[(2R)-pyrrolidin-2-yl]-1H-1,2,4-triazol-1-yl]pyridine
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-methanesulfonyl-N,2-dimethylpyrimidin-4-amine
6-[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S)-N-(3-benzylphenyl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
4-ethyl-1-(4-hydroxybutyl)-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-ethoxy-4-({4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(pyridin-3-yl)ethan-1-one
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[2-(propan-2-yloxy)ethyl]acetamide
2-methyl-6-{1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
N,N-dimethyl-5-({methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}methyl)pyrimidin-2-amine
2-[1-(3-methanesulfonamido-4-methoxyphenyl)-1H-imidazol-2-yl]benzoic acid
(2R,6R)-4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-(3-fluoropyridin-4-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine