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3-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
2,3,5,6-tetramethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]benzamide
7-[4-(benzyloxy)butanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
3-ethoxy-1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
8-fluoro-2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}quinoline
4-[3-(methylsulfanyl)butyl]-1-(2-phenylethyl)piperazin-2-one
2-[2-(2-methyl-1-benzofuran-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]acetic acid
8-methoxy-N-methyl-N-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}(methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(1-phenylcyclohexanecarbonyl)pyrrolidin-3-yl]methanol
[(2-fluorophenyl)methyl](2-methoxyethyl)(pyridin-4-ylmethyl)amine
2-(4-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
4-hydroxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
2-{[2-(difluoromethoxy)phenyl]methyl}-8-methyl-2,8-diazaspiro[4.5]decan-3-one
4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(piperidin-1-yl)butanamide
N-{4-[1-(4-sulfamoylphenyl)-1H-imidazol-2-yl]phenyl}acetamide
N-[2-(diethylamino)ethyl]-N-ethyl-5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(morpholin-4-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-cycloheptyl-2,3-dihydro-1H-inden-2-amine
1-(3-methyl-1H-pyrazole-5-carbonyl)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(1-phenylbutyl)oxane-4-carboxamide
ethyl 5-[(2,6-difluorophenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2,5-dimethyl-1-phenyl-1H-pyrrole
6-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-[(3R,4S)-1-(2-ethoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-4-(hydroxymethyl)benzamide
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-cyclopentyl-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,4-diazepan-6-ol
3-(4-chloro-2-methylbenzoyl)-1-(3,4,5-trimethoxybenzoyl)piperidine
(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-methyl-2-[N-methyl-1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanamide
2-cyclopropyl-5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]pyrimidin-4-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(methoxymethyl)-N-(pyridin-3-ylmethyl)cyclobutane-1-carboxamide
N-[(5-{[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}-3-methyl-1H-pyrazole-5-carboxamide
6,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(2-methylpiperidine-1-carbonyl)quinoline
3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
(3S,4S)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-(morpholin-4-yl)pyrrolidin-3-ol
5,6-dimethyl-2-[2-({4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}methyl)phenyl]-3,4-dihydropyrimidin-4-one
3-ethyl-1-[(5-fluoro-2-methoxyphenyl)methyl]piperidine-3-carboxylic acid
8-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1-oxa-8-azaspiro[4.5]decane
{2-[5-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}urea
1-[4-(1-hydroxy-2-methylpropyl)piperidin-1-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
3-methyl-2-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}pyridine
2-cyclopropanecarbonyl-8-(4-methoxy-2-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3R,5S)-N-cyclohexyl-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-methyl-3-[(2,3,6-trifluorophenyl)methyl]-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-4-(methylsulfanyl)benzamide
1-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}-1,4-diazepan-5-one