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5-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
N-(2-oxopyrrolidin-3-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
6-fluoro-N-[2-(5-methylfuran-2-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[ethyl({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
(4aR,8aR)-2-cyclopentanecarbonyl-7-{[3-(2-hydroxyethoxy)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,5-dichlorophenyl)urea
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(2-methylbutyl)piperidin-4-yl]imidazolidine-2,4-dione
(4aS,7aR)-1-[(2-methoxy-3,5-dimethylphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-(2-methoxyethyl)-5-methyl-3-phenyl-N-(1,3-thiazol-2-ylmethyl)-1,2-oxazole-4-carboxamide
1-(2-methoxypyridine-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
3-methoxy-2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}pyridine
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-4-(5-methylfuran-2-yl)benzamide
N-methyl-N-[4-(2-{[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}acetamido)phenyl]acetamide
1-[4-(4-hydroxyphenyl)piperazin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
3-{[(1-ethylcyclopropyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(pyrazin-2-yl)propan-1-one
(4-{5-[2-(furan-2-yl)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
2-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-N-[2-(4-methoxyphenyl)ethyl]acetamide
2-[(2-chlorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(2-methylphenoxy)-1-[2-(1H-pyrrol-1-yl)propanoyl]piperidine-4-carboxylic acid
2-(3-fluorophenyl)-1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidine
4-(dimethyl-1,3-thiazol-5-yl)-1H-indole
N-(2-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-oxoethyl)acetamide
N-(4-{2,7-diazaspiro[4.5]decane-7-carbonyl}phenyl)-2-(dimethylamino)acetamide
1,5-dimethyl-4-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(3S,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-[(2R,3R,6R)-5-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-({1-[2-(ethylamino)pyrimidine-5-carbonyl]piperidin-3-yl}methyl)-4-fluorobenzamide
({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)(pyridin-2-ylmethyl)amine
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4-(3-phenylpropyl)piperazin-2-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(2-hydroxypropyl)-1H-pyrazole-4-carboxamide
(3S,4S)-1-[(2-propylpyrimidin-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]propan-1-one
2-[4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]-1-(4-methylpiperidin-1-yl)ethan-1-one
{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}(methyl){[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
2-{[4-(2-amino-6-methoxypyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(5-methoxypyrimidin-2-yl)pyrrolidin-3-yl]methanol
4-methoxy-1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine
2-(azepan-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
{[3-(4-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[1-(3-methylpyridin-2-yl)ethyl]amine
3-[4-(3-hydroxyphenyl)piperidin-1-yl]-1-(3-methylpiperidin-1-yl)propan-1-one
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](methyl){[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
(3S,9aR)-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-methylphenyl)-5-(3-propoxypiperidine-1-carbonyl)pyrimidin-4-ol
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]acetamide
1-[2-(piperidin-2-yl)ethyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane