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1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)butan-1-one
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-phenylazepane
4-ethyl-3-(1-{3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
N,N-dimethyl-5-({4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}methyl)pyrimidin-2-amine
1-[4-(dimethyl-1,2-oxazol-4-yl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
N-{3-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-oxopropyl}-2-fluorobenzamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
1-[5-(dimethylamino)-2-methylphenyl]-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
(2R,3R)-3-[ethyl(methyl)amino]-1'-(6-methylpyridine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[4-(4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidin-1-yl)piperidin-1-yl]-1,3-benzoxazole
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(4aS,7aR)-1-(5-ethylthiophene-3-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzoxadiazole
4-{[(5-chlorothiophen-2-yl)methyl]amino}-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
2-{4-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-methyl-1,4-dihydroquinolin-4-one
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(oxan-4-yl)piperazine
2-(5-hydroxypyrazine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(pyridin-3-yl)-4-(1,3-thiazol-2-ylmethyl)morpholine
N-tert-butyl-9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-cyclopropyl-4-methoxy-3-({[(1S)-1-(3-methylpyridin-2-yl)ethyl]carbamoyl}amino)benzamide
4-[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]-N-phenylpiperidine-1-carboxamide
1-{3-[3-(2-chlorophenoxy)azetidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
(2H-1,3-benzodioxol-4-ylmethyl)[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amine
1-[(3-ethoxyphenyl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
3-{4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}-1-azabicyclo[2.2.2]octane
N-ethyl-2,7-dimethyl-N-[2-(phenylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidine-5-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
N,1-dimethyl-2-(morpholin-4-yl)-N-[1-(pyridin-3-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yloxy)acetamide
N-methyl-2,3-dioxo-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}cyclopropanecarboxamide
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-[(3-chloropyridin-4-yl)methyl]-4-(2-methoxyphenyl)-2-methylpiperazine
2,8-dimethyl-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]quinoline
5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyridin-2-amine
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-6-ethyl-1,2-dihydropyridin-2-one
2-[(4-chlorophenyl)methyl]-N-(oxolan-3-yl)-1,3-benzoxazole-5-carboxamide
4-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1-ethyl-1H-pyrrole-2-carbonitrile
(3-benzyl-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methanol
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1-methylcyclopropyl)propan-1-one
N-{3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}naphthalene-2-sulfonamide
(3aR,6aR)-2-(6-ethyl-2-methylpyrimidin-4-yl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid