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methyl 8-(cyclohex-3-en-1-ylmethyl)-1-[(3-methoxyphenyl)methoxy]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(1R,5S,6R)-3-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-(2-fluorophenoxymethyl)piperidine
4-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzene-1-sulfonamide
N-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
N-[2-({[4-(butan-2-yloxy)-3-chlorophenyl]methyl}amino)ethyl]methanesulfonamide
N-(3,5-dimethoxyphenyl)-3-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]propanamide
6-{1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){2-phenyl-1-[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]ethyl}amine
4-{1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-2-yl}quinoline
3-{[(2-methoxy-6-methylphenyl)carbamoyl](methyl)amino}-N-methylbutanamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
2-[3-(4-cyanopiperidine-1-carbonyl)benzenesulfonamido]-N,N-dimethylacetamide
4-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-pyrazol-4-yl)butan-1-one
3-methyl-N-[4-(5-methylfuran-3-amido)phenyl]-1-propyl-1H-pyrazole-4-carboxamide
(2S,4S)-4-amino-N-cyclopentyl-N-[(2,3-dimethoxyphenyl)methyl]-1-methylpyrrolidine-2-carboxamide
3-(2,5-difluorophenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]propan-1-one
1-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
(4aS,8aR)-6-(dimethyl-1,3-oxazole-5-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-({[(4-fluorophenyl)methyl](methyl)amino}methyl)-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
[1-(5-{[(5-methylthiophen-2-yl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
5-methyl-3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2-oxazole
methyl 1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
(1R,3S)-3-ethoxy-7-(2-methoxybenzenesulfonyl)-7-azaspiro[3.5]nonan-1-ol
2-cyclopentyl-N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[2-(dimethylamino)ethyl]acetamide
N-(2-{1-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}quinolin-6-yl)acetamide
2-[(5-{[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]methyl}pyrimidin-2-yl)(methyl)amino]acetic acid
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-5-phenyl-1,2-oxazole-3-carboxamide
3-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}benzonitrile
1-({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-2-ol
[(4aS,8aR)-6-(7-chloroquinolin-4-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
1-cyclohexyl-5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
7-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[2-(2,4-difluorophenyl)-1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
4-methyl-5-{[4-(1-phenylethyl)-1H-1,2,3-triazol-1-yl]methyl}-1,2,3-thiadiazole
1-(cyclohexylmethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-benzyl-4-oxo-5-(4-phenylpiperazine-1-carbonyl)-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N'-(2-fluoro-5-methylphenyl)butanediamide
N-ethyl-4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[2-(phenylsulfanyl)ethyl]benzamide
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
1-{6-hydroxy-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4-diazepan-1-yl}ethan-1-one
3-{1-[2-(2,4-dimethoxyphenyl)acetyl]piperidin-3-yl}benzoic acid
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-(2,3-difluorophenyl)-5-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
6-[4-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)piperidin-1-yl]-2-(propan-2-yl)pyrimidin-4-ol
8-[4-(1H-imidazol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-ethyl-N-[(2-fluorophenyl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(1S,2S)-2-[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]cyclohexan-1-ol