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3-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methylpyridine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(propan-2-yloxy)propanamide
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,2-dimethylpropanamide
4-{[1-(1-ethyl-6-oxopiperidine-3-carbonyl)azetidin-3-yl]oxy}benzoic acid
4-{5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl}pyridine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(2,4-dimethoxyphenyl)methyl]pyrrolidin-3-yl]methanol
1-ethyl-N-[(1-propylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
1-[(3R,4S)-3-(dimethylamino)-4-phenylpyrrolidin-1-yl]-3-methylbut-2-en-1-one
1-(cyclopropylmethyl)-N-methyl-5-(2-phenoxyacetyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(2-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)-4H-1,2,4-triazole
butyl 2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxylate
N-ethyl-N-methyl-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
1-{2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
2-amino-4-(4-fluoro-3-methoxyphenyl)-6-(furan-2-yl)pyridine-3-carbonitrile
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[2-(2-oxopyrrolidin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-amino-4-{methyl[2-(oxan-2-yl)ethyl]amino}quinazoline-6-carboxylic acid
{1-[(1-ethyl-1H-indol-3-yl)methyl]-3-[(4-fluorophenyl)methyl]piperidin-3-yl}methanol
7,8-dimethyl-3-[1-(pyridin-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-(4-methyl-3-phenylpiperazin-1-yl)-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
2-(but-3-enoyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2-chloro-4-fluorophenyl)-1-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
4-[(2,5-difluorophenyl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(pyridin-4-yl)propanamide
7-fluoro-2-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]quinoline-4-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(pyridine-2-carbonyl)morpholine
(2S)-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-2-phenylpiperazine
(3S,4S)-1-(6-methoxypyrimidin-4-yl)-4-propylpyrrolidine-3-carboxylic acid
7-[(2,3-difluorophenyl)methyl]-2-(2-methylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-[1-(4-methylpiperidine-4-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
(2S,4S)-1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-amino-N,N-diethylpyrrolidine-2-carboxamide
2-[5-(2-fluoro-4-methylphenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
4-(4-ethoxy-3-methylphenyl)-N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]butanamide
1-[1-ethyl-5-(5-propyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-(3-hydroxy-2,2-dimethylpropyl)-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
N,1-dimethyl-N-(1,2-oxazol-5-ylmethyl)-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(furan-2-ylmethyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]piperidine-4-carboxamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
3-propyl-1-[3-(pyridin-4-yl)propanoyl]piperidine-3-carboxylic acid
8-[(2-ethylpyrimidin-5-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-3-methylbut-2-en-1-one
({1-[(4-methoxyphenyl)methyl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl}methyl)urea
4-(2-chloro-4-fluorobenzoyl)-6-methoxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{4-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
7-(cyclopropylmethyl)-2-[2-(4H-1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-methyl-3-(pyridin-3-ylmethyl)-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-1-({4-[3-(dimethylcarbamoyl)pyridin-2-yl]phenyl}methyl)pyrrolidine-2-carboxylic acid
1-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)cyclopropane-1-carbonitrile
4-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]-N,N-dimethylaniline