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2-{1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-pyrazol-4-yl}ethan-1-ol
2-methyl-6-{1-[4-methyl-3-(1H-pyrrol-1-yl)benzoyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
2-(2-aminoethyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]quinazolin-4-amine
2-methyl-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
2-(dimethylamino)-7-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzene-1-sulfonamide
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[1-(thiophen-2-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide
3-[(4-{[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}piperidin-1-yl)methyl]phenol
1-(2-{[(4-phenyl-1,3-thiazol-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
2-(4-{6-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}phenoxy)ethan-1-ol
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-4-carboxamide
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
ethyl 4-({[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amino}methyl)-1H-pyrazole-3-carboxylate
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(methylsulfanyl)acetamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1-[2-(thiophen-2-yl)ethyl]urea
(4aS,7aR)-1-(2-cyclopropylacetyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-chlorophenyl)-N-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
3-(4-chlorophenyl)-5-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
1-{2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-amino-4-(3-ethyl-1,2-oxazol-5-yl)-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
1-({4-methyl-5-[1-(3,3,3-trifluoropropyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
5-(3,5-dichlorophenyl)-1,2,3,4-tetrahydroisoquinoline
3-{[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenol
N-[(5-chlorothiophen-2-yl)methyl]-1-cycloheptyl-6-oxopiperidine-3-carboxamide
7-chloro-3,5-dimethyl-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
N-cyclopentyl-9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-[methyl(2-phenylethyl)amino]-N-[(3S)-piperidin-3-yl]-2,3-dihydro-1H-indene-2-carboxamide
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-1H-1,2,4-triazole-5-carboxamide
1-(2-methanesulfonylethyl)-4-phenyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1H-imidazole
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-(furan-2-ylmethyl)acetamide
1-ethyl-N-[2-(4-methoxyphenyl)ethyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{1-[5-(morpholine-4-carbonyl)furan-2-yl]-1H-1,3-benzodiazol-2-yl}propan-1-ol
N-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-4-(2,2,2-trifluoroethyl)piperazine-1-carboxamide
methyl 3-(cyclobutylmethoxy)-5-(4-hydroxypiperidine-1-carbonyl)benzoate
1-(cyclohex-3-ene-1-carbonyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
3-{1-[5-(4-methoxyphenyl)furan-2-carbonyl]azetidin-3-yl}pyridine
N-butyl-N-methyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1-{7-[(3-ethoxy-4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]ethan-1-one
7-[(4-methoxy-2,5-dimethylphenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-{4-[3-(1H-pyrazol-1-yl)propyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-{[5-methyl-2-(4-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-3-(thiophen-2-yl)propanamide
1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-2-(2H-indazol-2-yl)ethan-1-one
2-amino-6-(3-hydroxyphenyl)-4-(3-phenyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile