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(2S,4R)-1-benzyl-N,N-diethyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-(dimethylamino)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(2-methylphenyl)ethan-1-one
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(4-methoxyphenoxymethyl)piperidine
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1H-1,3-benzodiazole-2-carboxamide
4-(2-chlorobenzoyl)-1-(2-methylphenyl)piperazin-2-one
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-(4-methylphenoxymethyl)piperidine
N,N-diethyl-1-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-amine
4-{[4-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)furan-2-yl]methyl}morpholine
N-cyclopropyl-3-{5-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
8-(3-fluoro-5-methylphenyl)quinolin-4-amine
3-(4-chlorophenyl)-5-(2-methanesulfonylethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1R,2R,6S,7S)-4-{[2-methyl-5-(1,2-oxazol-5-yl)thiophen-3-yl]sulfonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-[2-(2-methoxy-5-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenoxy)ethyl]-3-(trifluoromethyl)benzene-1-sulfonamide
4-(1H-imidazol-2-yl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
2-{1-[(3-methylphenyl)methyl]-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazol-3-yl}acetamide
benzyl (7S,9aR)-6,9-dioxo-7-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-[1-(cyclohexylmethyl)-4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
4-(hydroxymethyl)-1-[3-(2-methylphenyl)benzoyl]piperidin-4-ol
4-{[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
[1-(2-methoxyphenyl)ethyl](methyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
(2S,4R)-4-amino-N,N-diethyl-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidine-2-carboxamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-(morpholine-4-carbonyl)pyridin-4-amine
2-[3-oxo-9-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
4-({1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidin-2-yl}methyl)morpholine
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4-phenylazepane-1-carboxamide
11-(5-methoxy-1H-indole-2-carbonyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
methyl 3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(1-phenylpyrrolidin-3-yl)-3-propoxypiperidine
1-(4-{[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenyl)imidazolidin-2-one
(4aR,7aS)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
[(dimethyl-1,3-thiazol-5-yl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-(4-methoxyphenyl)-2,2-dimethyl-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
(1-{furo[3,2-c]pyridin-4-yl}-4-(2-phenylethyl)piperidin-4-yl)methanol
1-benzyl-8-[(3-chloro-4-hydroxyphenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[4-(4-methylpiperazin-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
(2R)-2-methyl-1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazine
3-{[(4-fluorophenyl)methyl]amino}-N-methyl-N-(propan-2-yl)benzamide
2-[4-(hydroxymethyl)phenyl]-1-[4-(4-methoxyphenoxy)piperidin-1-yl]ethan-1-one
1-(1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)piperidin-4-ol
1-(furan-3-ylmethyl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(2,2,2-trifluoroethyl)pyrimidin-2-amine
6-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrazine-2-carboxylic acid
1-(2-methoxyethyl)-4-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}pyrrolidin-2-one
N-[1-(2,5-dimethoxyphenyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(3-methoxypropyl)-8-[2-(methylamino)pyridine-4-carbonyl]-2,8-diazaspiro[4.5]decan-3-one