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2-(2H-1,3-benzodioxol-5-yl)-1-[4-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]ethan-1-one
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
9-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(5-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}furan-2-yl)methanol
2-(methylsulfanyl)-3-[2-(pyridin-2-yl)piperidine-1-carbonyl]pyridine
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(3-methoxybenzoyl)piperidine
3-methyl-5-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1,2-oxazole
2-[methyl(piperidin-4-yl)amino]-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one
3-(1H-indol-3-yl)-1-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
ethyl({[2-(furan-2-yl)pyrimidin-5-yl]methyl}){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-propylpiperidine-1-carboxamide
3-{5-[2-(oxan-2-ylmethoxy)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-methyl-4-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
4-phenyl-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine-4-carbonitrile
4-[(2,2-difluoroethyl)sulfamoyl]-N-[3-(methylsulfanyl)propyl]benzamide
5-cyclopropyl-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-methyl-1H-pyrazole-4-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-(piperidin-3-yl)benzamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
N-benzyl-N-methyl-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
3-{[1-(4-cyanooxane-4-carbonyl)pyrrolidin-3-yl]methyl}benzamide
1-(2-methylpropyl)-4-[(3-methylquinoxalin-2-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-ethyl-5-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}pyrimidine
3-(3-hydroxy-3-methylbutyl)-N-[1-(1H-imidazol-2-yl)ethyl]benzamide
3-({1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
5-phenyl-4-[1-(2-phenylethyl)piperidin-3-yl]-2-(pyridin-4-yl)pyrimidine
2-(2-methylpropyl)-8-{[2-(methylsulfanyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
N-methyl-2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carboxamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrimidin-2-amine
N-[4-({[(5-methylpyrazin-2-yl)methyl]carbamoyl}methyl)phenyl]butanamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,2R,6S,7S)-4-(1,8-naphthyridine-2-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propane-1,3-diol
N-[(2-methylphenyl)(phenyl)methyl]-3-(2-oxopiperidin-1-yl)propanamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-4-(morpholin-4-yl)-N-(pyridin-3-ylmethyl)benzamide
N-methyl-N-(2-phenylethyl)-2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,3-dihydro-1H-inden-2-amine
2-ethyl-9-[5-(methoxymethyl)thiophene-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
8-[5-(1H-1,2,4-triazol-5-ylsulfanyl)furan-2-yl]-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-6-one
3,5-dimethoxy-2-({4-[(methylcarbamoyl)methyl]piperazin-1-yl}methyl)benzoic acid
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]furan-3-carboxamide
2-(3-fluorophenoxymethyl)-N-[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
2-amino-4-{2-[2-(dimethylamino)ethoxy]phenyl}-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
7-[4-(1H-pyrrol-1-ylmethyl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(pyridin-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-hydroxy-3-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}benzamide
4-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-9,10-dihydroacridin-9-one
2-[(3-chlorophenyl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
1-[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
4-(4-methylphenoxy)-1-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)piperidine-4-carboxylic acid