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2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}acetamide
1-({4-methyl-5-[1-(2-propoxyethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-phenoxy-N-(1-{[(prop-2-en-1-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)propanamide
9-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1,4,9-triazaspiro[5.5]undecan-5-one
{3-[(3-methoxyphenyl)methyl]-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl}methanol
3-(2-phenylethyl)-7-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-(piperidin-1-ylmethyl)-4-(5-propyl-1,2-oxazole-3-carbonyl)-1,4-oxazepane
5-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
1-[(2-fluorophenyl)methyl]-2-methyl-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidine-2-carboxamide
ethyl 5-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
8-(1-benzofuran-2-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propane-1,2-dione
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
3-fluoro-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyridine-4-carboxamide
5-methyl-1-[4-(4-{[(2R)-3-methylbutan-2-yl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
4-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-methyl-5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(piperidin-1-yl)pyrimidine
methyl 3-(pyridin-2-yl)benzoate
1-[1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl]piperidine-4-carbonitrile
N-(2-{[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}ethyl)acetamide
2-[(4-chlorophenyl)methyl]-8-(pyrrolidin-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}propanamide
5-(3,3-diphenylpiperidine-1-carbonyl)-2-methyl-1H-1,3-benzodiazole
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-phenylpropanamide
1-(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)ethan-1-one
2-({5-[1-methyl-3-(pyridin-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]furan-2-yl}sulfanyl)pyrimidine
3-cyano-N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]benzamide
7-(3-chlorophenyl)-4-(furan-3-carbonyl)-9-[(1-methylpiperidin-3-yl)methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(morpholine-4-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
2-(2-methoxy-4-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}phenoxy)acetamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-methoxy-N-methylpyrimidin-2-amine
N-(1,2-benzoxazol-6-yl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carboxamide
N-ethyl-2-(2-fluorophenoxymethyl)-N-(oxan-4-ylmethyl)-1,3-oxazole-4-carboxamide
6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
6-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}quinazolin-4-amine
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
dimethyl({5-[1-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1H-imidazol-2-yl]thiophen-3-yl}methyl)amine
2-methyl-6-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
6-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-phenyl-1-[4-(1,2,5-thiadiazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-1-ol
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-ethyl-N-[2-(morpholin-4-yl)ethyl]acetamide