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3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-1-[4-(methoxymethyl)piperidin-1-yl]propan-1-one
2-(4-ethyl-2,3-dioxopiperazin-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
ethyl 5-(1H-indole-3-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
1-[(3-methyl-1H-indol-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-[3-(4-benzoylpiperazin-1-yl)-3-oxopropyl]imidazolidine-2,4-dione
4-benzyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-2-one
N-(4-methoxyphenyl)-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-3-amine
N-cyclopropyl-N-[(4-hydroxyphenyl)methyl]spiro[2.2]pentane-1-carboxamide
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-N-(1,1,1-trifluoropropan-2-yl)-2,3-dihydro-1H-isoindole-4-carboxamide
3-{2-oxo-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
5-(phenoxymethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
4-(5-acetylthiophene-3-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyrrolidin-1-yl)ethan-1-one
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
N-methyl-5-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[2-(4H-1,2,4-triazol-4-yl)phenyl]acetamide
3-{[(4-fluorophenyl)methyl]amino}-N-[1-(1H-imidazol-1-yl)butan-2-yl]benzamide
3-{2-[3-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
N-ethyl-2-methyl-N-[3-(morpholin-4-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
1-cyclopropyl-5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}piperidin-2-one
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methyl-1,3-thiazole-4-carboxamide
(1S,5R)-6-(1,3-thiazol-4-ylmethyl)-3-[3-(thiophen-2-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
N-(2-{1-[(6-chloropyridin-3-yl)methyl]piperidin-3-yl}ethyl)methanesulfonamide
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
8-(2-aminoacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-5-(pyrrolidin-1-yl)pyridazine
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[2-(1H-1,2,4-triazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
5-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(1-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
6-ethyl-2-methyl-N-[2-(1,3-thiazol-4-yl)ethyl]quinoline-4-carboxamide
(3R,4R)-1-[(2-ethylpyrimidin-4-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-[2-(4-fluorobenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
1-(2,6-dimethoxypyridin-3-yl)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}urea
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
8-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(3-methylbut-2-enoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(2-{1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl}acetyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
1-ethyl-4-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]benzonitrile
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}quinoline-3-carboxamide
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(3-acetylbenzoyl)-1-(3,5-dimethylphenyl)piperazin-2-one
2-{5-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-1,3-benzodiazole
(2E)-N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
{5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]furan-2-yl}methanol
5-methoxy-1-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-indole-2-carboxamide