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1-[(3S)-3-ethylmorpholin-4-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
5-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
1-methyl-5-phenyl-N-[(3R)-piperidin-3-yl]-1H-pyrazole-3-carboxamide
(2-{[1-(1,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]oxy}ethyl)dimethylamine
3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-(5-methylpyridin-3-yl)benzamide
6-(2,5-dimethylfuran-3-yl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
3-{1-[3-(pyrrolidine-1-sulfonyl)thiophene-2-carbonyl]azetidin-3-yl}pyridine
methyl 1-[(3R,5S)-1-(3-methylbut-2-en-1-yl)-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(1,3-benzothiazol-2-ylmethyl)methylamine
2-methyl-1-[1-(2-methyl-1-benzofuran-5-carbonyl)azetidin-3-yl]piperidine
1-({1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-yl}amino)-3-(3-methoxyphenoxy)propan-2-ol
N-[(3R,5S)-1-cyclohexyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-5-ethyl-1,2-oxazole-3-carboxamide
1-(4-ethenylbenzoyl)-N-(4-methoxyphenyl)piperidin-3-amine
5-(dimethyl-1,3-thiazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-chloro-5-acetamido-N-(2-methylprop-2-en-1-yl)benzamide
2-({[1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
N-[4-(1-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-1,2,3-triazol-4-yl)phenyl]acetamide
N2-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N2,N4-dimethylpyrimidine-2,4-diamine
4-(4-benzyl-1H-pyrazol-5-yl)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidine
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]quinoxaline-6-carboxamide
{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
2-[1-(cyclohexylmethyl)-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl]ethan-1-ol
N-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-3-hydroxybenzamide
N-propyl-5-(1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(3-hydroxyphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-methoxy-1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
1-{2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)pyridine-3-carbonyl}piperidine-4-carboxamide
N-[(3S,4R)-1-(3-chlorothiophene-2-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
1-[2-(2,3-dimethylphenoxy)ethyl]-5-methylpyrrolidin-2-one
(4aS,7aR)-1-[3-(2-fluorophenyl)propanoyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)-6-methoxyphenol
ethyl 4-[(2-chlorophenyl)methyl]-1-(pyridine-3-sulfonyl)piperidine-4-carboxylate
1-[7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
2-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2,2-dimethyl-N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-methoxy-4-[(3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[2-hydroxy-4-(methylsulfanyl)butanoyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
(1R,3S)-3-(2-aminoethoxy)-7-(2,1,3-benzothiadiazol-5-ylmethyl)-7-azaspiro[3.5]nonan-1-ol
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
3-(hydroxymethyl)-1-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}piperidin-3-ol
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one