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5-[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-[(3S,4R)-1-(2-methylpropyl)-4-(morpholin-4-yl)piperidin-3-yl]-N-[2-(morpholin-4-yl)ethyl]propanamide
3-{5-[(4-methyl-1,3-thiazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(morpholin-4-yl)propan-1-one
3-(2-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-2-oxoethyl)-1,3-thiazolidine-2,4-dione
2-(2,4-dimethoxy-3-methylphenyl)-4-[(2,4-dimethyl-1H-imidazol-1-yl)methyl]-5-methyl-1,3-oxazole
1-ethyl-3-(propan-2-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
1-(2-chlorobenzoyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
2-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{2-[(1H-indol-4-ylmethyl)amino]pyrimidin-4-yl}piperidin-4-ol
3-{2-[4-(2-methoxyethoxy)piperidin-1-yl]-2-oxoethyl}-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-one
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}pyridine-3-carbonitrile
[(2,4-dimethoxyphenyl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-[2-(ethylsulfanyl)ethyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(2S)-pyrrolidine-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-ethyl-5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
5-benzyl-3-[2-(pyrrolidin-1-yl)ethyl]-5-[1-(thiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperidine
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
5-(methoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-3-methyl-1-[3-(1,3-oxazol-5-yl)phenyl]urea
2-[1-(thiophene-2-sulfonyl)pyrrolidin-2-yl]pyridine
2-(5-methyl-2-oxo-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperazin-1-yl)benzonitrile
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-({1-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-N-(propan-2-yl)acetamide
N-[(3R,4R)-3-hydroxy-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyridine-2-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[methyl(2-phenylethyl)amino]methyl}piperidin-2-one
3-tert-butyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,2,4-triazole
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-3-(3-methylphenyl)-1H-pyrazole
3-{1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-1-propyl-1H-pyrazole-5-carboxamide
7-(cyclopropylmethyl)-2-[1-(3-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
1-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethan-1-one
(2S,4R)-4-amino-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-methylpyrrolidine-2-carboxamide
3-{2-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}acetic acid
N-cyclohexyl-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-tert-butyl-4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carboxamide
4-ethyl-3-{[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
(3R,4R)-1-[(4-fluoro-2-methoxyphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
N-(cyclohexylmethyl)-3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(4-fluorophenyl)methyl]-1,1-dioxo-N-(pyridin-4-ylmethyl)-1λ6-thiolane-3-carboxamide
N-[1-(4-methanesulfonylphenyl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-cyclobutanecarbonyl-9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
methyl 1-(2-methoxyethyl)-5-{[(2E)-2-methylbut-2-en-1-yl]amino}-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate