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6-methyl-2-(4-methylphenoxymethyl)-1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridin-4-one
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(2-methoxyphenyl)propanamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-phenoxybenzamide
6-ethyl-2-methyl-4-[2-(1-methyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]quinoline
3-{[2-(difluoromethoxy)phenyl]methyl}-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2S)-N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-acetamidopropanamide
2-cyclopentyl-1-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
(4S)-1-[(6-ethoxypyridin-3-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
8-[(3-chloro-4-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
6-{[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}-1-methyl-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one
1-(2-methoxy-6-methylphenyl)-3-methyl-3-[(4-methyl-1H-imidazol-2-yl)methyl]urea
1-benzyl-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-acetamido-2-methyl-1H-1,3-benzodiazole-7-carboxamide
({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)[2-(1H-imidazol-1-yl)ethyl]methylamine
N-(2-methoxyethyl)-1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
1-methyl-5-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2-methoxyphenyl)methyl]-N3-(1-methoxypropan-2-yl)-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
N-{[1-(2-acetamidoacetyl)piperidin-3-yl]methyl}-4-fluorobenzamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(3-phenyl-1,2-oxazole-4-carbonyl)piperidine
3-(2-chlorophenyl)-1-(morpholin-4-yl)-3-phenylpropan-1-one
N-(3-hydroxyadamantan-1-yl)-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
(2S,4R)-1-[(2,5-dimethylphenyl)methyl]-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
ethyl 2-(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)acetate
2-(2H-1,2,3-benzotriazol-2-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
5-({4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)-2-methylpyrimidine
2-[5-(2,2-dimethyloxan-4-yl)-1-methyl-1H-1,2,4-triazol-3-yl]pyridine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[4-(piperidin-1-yl)benzoyl]piperidin-3-ol
methyl 5-{7-[(3,4-difluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-5-oxopentanoate
6-[(3-methoxyphenyl)methyl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
6-[(2E)-3-(3,5-difluorophenyl)prop-2-enoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
({2-[(2-chloroprop-2-en-1-yl)oxy]-7-fluoroquinolin-3-yl}methyl)[3-(1H-imidazol-1-yl)propyl]amine
1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-4-(thiophen-2-yl)butan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-N,2,6-trimethylpyrimidine-4-carboxamide
N-[2-(5-methylfuran-2-yl)ethyl]-4-sulfamoylbenzamide
3-{4-[(6-chloro-2H-chromen-3-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
2,5-dimethyl-3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrazine
2-[(4aR,7aS)-4-[(2,6-dimethylphenyl)carbamoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
methyl (2S)-2-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-1,2-oxazol-5-yl]formamido}-3-phenylpropanoate
(4aR,7aS)-1-acetyl-4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-3-{5-[2-methyl-2-(morpholin-4-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
7-[(2,3-dimethoxyphenyl)methyl]-2-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
4-(4-fluorophenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-acetyl-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
4-[(6-methylpyridin-3-yl)oxy]-1-{[(1s,4s)-4-aminocyclohexyl]methyl}piperidine-4-carboxylic acid
6-(2-chlorophenyl)-N,N,7-trimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
9-methoxy-7-(5-methylthiophen-2-yl)-4-[2-(pyridin-2-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl (2S)-2-{[5-(2,6-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}-2-phenylacetate