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2-(3-chlorophenyl)-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]acetamide
methyl 3-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}propanoate
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-hydroxyethyl)-N-methylbenzamide
1'-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N,2-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-1H-pyrrole-3-carboxamide
7-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-phenylphenyl)piperazin-2-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[(3,4,5-trimethoxyphenyl)methyl]piperidine-3-carboxamide
5-{2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-methyl-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]urea
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methylpropanamide
1-[4-({4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
3-{[1-(3,4-difluorophenyl)piperidin-4-yl](methyl)amino}-N-methylpropanamide
6-(adamantane-1-carbonyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
5-(1-ethyl-1H-imidazol-5-yl)-1-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-phenyl-1H-imidazole
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide
{4-[(1-benzyl-1H-indol-6-yl)methyl]-1-methylpiperazin-2-yl}methanol
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-(1H-indol-3-yl)pyridine-3-carbonitrile
1-methyl-4-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
6-(2-phenylethyl)-2-[3-(piperazin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-{2-[4-(trifluoromethyl)phenyl]ethyl}-1,2-oxazole-5-carboxamide
4-hydroxy-2-methyl-N-[1-(thiophen-3-yl)propan-2-yl]pyrimidine-5-carboxamide
1-[(1-methyl-1H-indol-5-yl)methyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
1-{3-[3-(3-methylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-[2-(3-fluorophenyl)-2-hydroxyethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
3-[(3,4-dimethoxyphenyl)methyl]-5-[(2-ethyl-4-methyl-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
(3S,7S)-5-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
(3S,4R)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
2-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-(trifluoromethyl)pyridine
N-cyclopropyl-5-[(4-oxo-4H-chromen-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
2-[(3,4-difluorophenyl)methyl]-8-[(2R)-pyrrolidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-[4-(4-{[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
3-(4-chlorophenyl)-3-phenyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
5-{[4-(4-propyl-1,4-diazepane-1-carbonyl)-1,3-oxazol-2-yl]methoxy}isoquinoline
8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](isoquinolin-5-ylmethyl)methylamine
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-4-(pyridin-2-yl)pyrimidin-2-amine
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-2-(morpholin-2-yl)acetamide
3-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propanoic acid
1-cyclopentyl-N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-1H-pyrazol-5-amine
1-[(2,3-difluorophenyl)methyl]-5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
1-(2-chlorophenyl)-3-{1-[1-(3-fluoropropyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-(cyclopropylmethyl)-3-{methyl[(2-methylpyridin-4-yl)methyl]sulfamoyl}benzamide
dimethyl[2-(2-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)ethyl]amine
3-{5-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
(3S)-1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carbonyl}pyrrolidin-3-ol
2-{2-[3-(3-methylpiperazine-1-carbonyl)benzenesulfonamido]ethoxy}ethan-1-ol