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2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N-methylpyridine-4-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[2-(pyridin-3-yl)ethyl]butanamide
(2E)-N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylbut-2-enamide
4-{4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}morpholine
6-methyl-2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridine-3-carboxamide
7-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-(3-methoxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
2-methyl-6-(1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)pyrimidin-4-ol
4-methyl-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2,3-thiadiazole-5-carboxamide
(1S,5R)-3-(2-chloro-4-fluorobenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4S)-1-(dimethyl-1,3-oxazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
3-ethyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1-methyl-1H-pyrazole-5-carboxamide
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
(3aR,6aR)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-(1-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-methylpropan-2-yl)morpholine
(2R,6R)-4-[2-(2-oxopyrrolidin-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
3-[3-(heptan-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-6-methylpyridazine
5-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-2-cyclohexylpyrimidine
(1R,5S)-3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
[(2S,6S)-11-methoxy-4-(2-phenoxyethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(3S,4R)-3-benzyl-1-methyl-4-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]piperidine
4-[(4aS,8aR)-decahydroisoquinolin-2-yl]-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
2-cyclopropyl-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
2-[1-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]phenol
[(2S)-1-[2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carbonyl]pyrrolidin-2-yl]methanol
N,N,4-trimethyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
N-ethyl-6-fluoro-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
(3S,4R)-N,N-dimethyl-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-propylpyrrolidin-3-amine
3-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
3-(furan-2-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
1-(2,3-dimethylphenyl)-3-methyl-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]urea
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{[1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
1-[1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidin-4-ol
4-(1-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}-2-methylpropan-2-yl)morpholine
N-methyl-2-(pyridin-3-yl)-N-(pyrimidin-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{2-[2-(trifluoromethyl)phenyl]ethyl}propanamide
N,N-diethyl-1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidine-3-carboxamide
2-({4-phenyl-5-[1-(propan-2-yloxy)ethyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
4-[(3-methylphenyl)methyl]-1-(4-oxo-4H-chromene-2-carbonyl)-1,4-diazepan-5-one
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-3-(piperidin-3-yl)benzamide
1-tert-butyl-5-(methoxymethyl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazole
2-[(4-chlorophenyl)methyl]-8-(2,6-diaminopyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
4-methyl-N-(2-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
4-({1-[(propan-2-yloxy)carbonyl]pyrrolidin-3-yl}methyl)benzoic acid
8-fluoro-2-({[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}methyl)quinolin-4-ol
2-(adamantan-1-yl)-N-(2,3-dihydroxypropyl)-N-methylacetamide
1-(4-methoxyphenyl)-4-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperazin-2-one
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-3-propanamidobenzamide